[Gastrointestinal Spice Sensors and Their Functions].
Horie, Syunji; Tashima, Kimihito; Matsumoto, Kenjiro.
; 138(8): 1003-1009, 2018.
Artigo em Japonês | MEDLINE | ID: mdl-30068839
Medicinal Chemistry, Pharmacology, and Clinical Implications of TRPV1 Receptor Antagonists.
Rational design and validation of a vanilloid-sensitive TRPV2 ion channel.
Involvement of the TRPV1 channel in the modulation of spontaneous locomotor activity, physical performance and physical exercise-induced physiological responses
Understanding TRPV1 activation by ligands: Insights from the binding modes of capsaicin and resiniferatoxin.
Carboxyl-terminal domain of transient receptor potential vanilloid 1 contains distinct segments differentially involved in capsaicin- and heat-induced desensitization.
Binding of Capsaicin to the TRPV1 Ion Channel.
Tris-hydroxymethyl-aminomethane enhances capsaicin-induced intracellular Ca(2+) influx through transient receptor potential V1 (TRPV1) channels.
Quantitative characterization of capsaicin-induced TRPV1 ion channel activation in HEK293 cells by impedance spectroscopy.
α-Substituted 2-(3-fluoro-4-methylsulfonamidophenyl)acetamides as potent TRPV1 antagonists.
TRPV1 channels and the progesterone receptor Sig-1R interact to regulate pain.