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Trioxolane-Mediated Delivery of Mefloquine Limits Brain Exposure in a Mouse Model of Malaria.
Lauterwasser, Erica M W; Fontaine, Shaun D; Li, Hao; Gut, Jiri; Katneni, Kasiram; Charman, Susan A; Rosenthal, Philip J; Bogyo, Matthew; Renslo, Adam R.
Affiliation
  • Lauterwasser EM; Department of Pharmaceutical Chemistry and Department of Medicine, University of California San Francisco , 1700 Fourth Street, San Francisco, California 94158, United States.
  • Fontaine SD; Department of Pharmaceutical Chemistry and Department of Medicine, University of California San Francisco , 1700 Fourth Street, San Francisco, California 94158, United States.
  • Li H; Departments of Pathology and Microbiology and Immunology, Stanford School of Medicine , 300 Pasteur Drive, Stanford, California 94305, United States.
  • Gut J; Department of Pharmaceutical Chemistry and Department of Medicine, University of California San Francisco , 1700 Fourth Street, San Francisco, California 94158, United States.
  • Katneni K; Centre for Drug Candidate Optimisation, Monash Institute of Pharmaceutical Sciences, Monash University , Parkville, VIC 3052, Australia.
  • Charman SA; Centre for Drug Candidate Optimisation, Monash Institute of Pharmaceutical Sciences, Monash University , Parkville, VIC 3052, Australia.
  • Rosenthal PJ; Department of Pharmaceutical Chemistry and Department of Medicine, University of California San Francisco , 1700 Fourth Street, San Francisco, California 94158, United States.
  • Bogyo M; Departments of Pathology and Microbiology and Immunology, Stanford School of Medicine , 300 Pasteur Drive, Stanford, California 94305, United States.
  • Renslo AR; Department of Pharmaceutical Chemistry and Department of Medicine, University of California San Francisco , 1700 Fourth Street, San Francisco, California 94158, United States.
ACS Med Chem Lett ; 6(11): 1145-9, 2015 Nov 12.
Article in En | MEDLINE | ID: mdl-26617969

Full text: 1 Collection: 01-internacional Database: MEDLINE Language: En Journal: ACS Med Chem Lett Year: 2015 Document type: Article Affiliation country: United States Country of publication: United States

Full text: 1 Collection: 01-internacional Database: MEDLINE Language: En Journal: ACS Med Chem Lett Year: 2015 Document type: Article Affiliation country: United States Country of publication: United States