Detalhe da pesquisa
1.
Discovery of 2-amino-3-amido-5-aryl-pyridines as highly potent, orally bioavailable, and efficacious PERK kinase inhibitors.
Bioorg Med Chem Lett;
43: 128058, 2021 07 01.
Artigo
em Inglês
| MEDLINE
| ID: mdl-33895276
2.
Discovery of HC-7366: An Orally Bioavailable and Efficacious GCN2 Kinase Activator.
J Med Chem;
67(7): 5259-5271, 2024 Apr 11.
Artigo
em Inglês
| MEDLINE
| ID: mdl-38530741
3.
Discovery and optimization of 7-aminofuro[2,3-c]pyridine inhibitors of TAK1.
Bioorg Med Chem Lett;
23(16): 4517-22, 2013 Aug 15.
Artigo
em Inglês
| MEDLINE
| ID: mdl-23850198
4.
Novel 6-aminofuro[3,2-c]pyridines as potent, orally efficacious inhibitors of cMET and RON kinases.
Bioorg Med Chem Lett;
23(15): 4381-7, 2013 Aug 01.
Artigo
em Inglês
| MEDLINE
| ID: mdl-23773865
5.
Optimization of a Novel Mandelamide-Derived Pyrrolopyrimidine Series of PERK Inhibitors.
Pharmaceutics;
14(10)2022 Oct 19.
Artigo
em Inglês
| MEDLINE
| ID: mdl-36297668
6.
OSI-930: a novel selective inhibitor of Kit and kinase insert domain receptor tyrosine kinases with antitumor activity in mouse xenograft models.
Cancer Res;
66(2): 1015-24, 2006 Jan 15.
Artigo
em Inglês
| MEDLINE
| ID: mdl-16424037
7.
Dihydropyridines as inhibitors of capacitative calcium entry in leukemic HL-60 cells.
Biochem Pharmacol;
65(3): 329-38, 2003 Feb 01.
Artigo
em Inglês
| MEDLINE
| ID: mdl-12527326
8.
Preparation of Enantiomerically Enriched (2R,3R)- or (2S,3S)-trans-2,3-Diaryloxiranes via Camphor-Derived Sulfonium Ylides.
J Org Chem;
61(2): 489-493, 1996 Jan 26.
Artigo
em Inglês
| MEDLINE
| ID: mdl-11666965
9.
A Direct Route to C-Vinylaziridines: Reaction of N-Sufonylimines with Allylic Ylides under Phase-Transfer Conditions or with Preformed Ylides at Low Temperature.
J Org Chem;
61(14): 4641-4648, 1996 Jul 12.
Artigo
em Inglês
| MEDLINE
| ID: mdl-11667392
10.
A3 Adenosine Receptors: Protective vs. Damaging Effects Identified Using Novel Agonists and Antagonists.
Drug Dev Res;
45(3-4): 113-124, 1998.
Artigo
em Inglês
| MEDLINE
| ID: mdl-31808655
11.
Pyran Template Approach to the Design of Novel A3 Adenosine Receptor Antagonists.
Drug Dev Res;
48(4): 171-177, 1999 Dec.
Artigo
em Inglês
| MEDLINE
| ID: mdl-27182099
12.
Asymmetric Ylide Reactions: Epoxidation, Cyclopropanation, Aziridination, Olefination, and Rearrangement.
Chem Rev;
97(6): 2341-2372, 1997 Oct 01.
Artigo
em Inglês
| MEDLINE
| ID: mdl-11848902
13.
Discovery of an Orally Efficacious Imidazo[5,1-f][1,2,4]triazine Dual Inhibitor of IGF-1R and IR.
ACS Med Chem Lett;
1(9): 510-5, 2010 Dec 09.
Artigo
em Inglês
| MEDLINE
| ID: mdl-24900240
14.
A highly effective one-pot synthesis of quinolines from o-nitroarylcarbaldehydes.
Org Biomol Chem;
5(1): 61-4, 2007 Jan 07.
Artigo
em Inglês
| MEDLINE
| ID: mdl-17164907