Detalhe da pesquisa
1.
Discovery of berberine analogs as potent and highly selective p300/CBP HAT inhibitors.
Bioorg Chem;
138: 106597, 2023 09.
Artigo
em Inglês
| MEDLINE
| ID: mdl-37245245
2.
Design, synthesis, and antitumor study of a series of novel 1-Oxa-4-azaspironenone derivatives.
Bioorg Med Chem Lett;
74: 128925, 2022 10 15.
Artigo
em Inglês
| MEDLINE
| ID: mdl-35944852
3.
Design, synthesis, and antitumor activity evaluation of novel acyl sulfonamide spirodienones.
Bioorg Med Chem;
60: 116626, 2022 04 15.
Artigo
em Inglês
| MEDLINE
| ID: mdl-35255412
4.
One-Pot Synthesis of Seven-Membered Heterocyclic Derivatives of Diazepines Involving Copper-Catalyzed Rearrangement Cascade Allyl-Amination.
J Org Chem;
85(8): 5146-5157, 2020 04 17.
Artigo
em Inglês
| MEDLINE
| ID: mdl-32182067
5.
Development of a bioavailable boron-containing PI-103 Bioisostere, PI-103BE.
Bioorg Med Chem Lett;
30(14): 127258, 2020 07 15.
Artigo
em Inglês
| MEDLINE
| ID: mdl-32527558
6.
Novel one-pot synthesis of imidazolinones from esters: a concise synthesis of GSK2137305.
Org Biomol Chem;
18(11): 2175-2181, 2020 03 18.
Artigo
em Inglês
| MEDLINE
| ID: mdl-32147677
7.
Design, Synthesis, and Antitumor Activity of a Series of Novel 4-(Aromatic Sulfonyl)-1-oxa-4-azaspiro[4.5]deca-6,9-dien-8-ones.
Molecules;
25(22)2020 Nov 21.
Artigo
em Inglês
| MEDLINE
| ID: mdl-33233396
8.
Synthesis and antiproliferative evaluation of new zampanolide mimics.
Org Biomol Chem;
17(15): 3830-3844, 2019 04 10.
Artigo
em Inglês
| MEDLINE
| ID: mdl-30924817
9.
Nitrogen-containing derivatives of O-tetramethylquercetin: Synthesis and biological profiles in prostate cancer cell models.
Bioorg Chem;
87: 227-239, 2019 06.
Artigo
em Inglês
| MEDLINE
| ID: mdl-30904813
10.
Synthesis and Antitumor Activity of a Series of Novel 1-Oxa-4-azaspiro[4,5]deca-6,9-diene-3,8-dione Derivatives.
Molecules;
24(5)2019 Mar 07.
Artigo
em Inglês
| MEDLINE
| ID: mdl-30866506
11.
Optimization of diarylpentadienones as chemotherapeutics for prostate cancer.
Bioorg Med Chem;
26(16): 4751-4760, 2018 09 01.
Artigo
em Inglês
| MEDLINE
| ID: mdl-30121214
12.
Optimized synthesis and antiproliferative activity of desTHPdactylolides.
Bioorg Med Chem;
26(12): 3514-3520, 2018 07 23.
Artigo
em Inglês
| MEDLINE
| ID: mdl-29784275
13.
O-Aminoalkyl-O-Trimethyl-2,3-Dehydrosilybins: Synthesis and In Vitro Effects Towards Prostate Cancer Cells.
Molecules;
23(12)2018 Nov 29.
Artigo
em Inglês
| MEDLINE
| ID: mdl-30501133
14.
3-O-Substituted-3',4',5'-trimethoxyflavonols: Synthesis and cell-based evaluation as anti-prostate cancer agents.
Bioorg Med Chem;
25(17): 4768-4777, 2017 09 01.
Artigo
em Inglês
| MEDLINE
| ID: mdl-28760528
15.
5- or/and 20-O-alkyl-2,3-dehydrosilybins: Synthesis and biological profiles on prostate cancer cell models.
Bioorg Med Chem;
25(17): 4845-4854, 2017 09 01.
Artigo
em Inglês
| MEDLINE
| ID: mdl-28756013
16.
Ligands of Therapeutic Utility for the Liver X Receptors.
Molecules;
22(1)2017 Jan 05.
Artigo
em Inglês
| MEDLINE
| ID: mdl-28067791
17.
A new class of flavonol-based anti-prostate cancer agents: Design, synthesis, and evaluation in cell models.
Bioorg Med Chem Lett;
26(17): 4241-5, 2016 09 01.
Artigo
em Inglês
| MEDLINE
| ID: mdl-27476422
18.
3-O-Alkyl-2,3-dehydrosilibinins: Two synthetic approaches and in vitro effects toward prostate cancer cells.
Bioorg Med Chem Lett;
26(14): 3226-3231, 2016 07 15.
Artigo
em Inglês
| MEDLINE
| ID: mdl-27261177
19.
Design, synthesis, and biological evaluation of 1,9-diheteroarylnona-1,3,6,8-tetraen-5-ones as a new class of anti-prostate cancer agents.
Bioorg Med Chem;
24(19): 4692-4700, 2016 10 01.
Artigo
em Inglês
| MEDLINE
| ID: mdl-27543391
20.
Discovery of Novel Allopurinol Derivatives with Anticancer Activity and Attenuated Xanthine Oxidase Inhibition.
Molecules;
21(6)2016 Jun 20.
Artigo
em Inglês
| MEDLINE
| ID: mdl-27331805