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Diamine Derivatives as Novel Small-Molecule, Potent, and Subtype-Selective Somatostatin SST3 Receptor Agonists.
Li, Derun; Wu, Zhicai; Yu, Yang; Ball, Richard G; Guo, Liangqin; Sherer, Edward; He, Shuwen; Hong, Qingmei; Lai, Zhong; Qi, Hongbo; Truong, Quang; Yang, David X; Chicchi, Gary G; Tsao, Kwei-Lan; Trusca, Dorina; Trujillo, Maria; Pachanski, Michele; Eiermann, George J; Howard, Andrew D; Zhou, Yun-Ping; Zhang, Bei B; Nargund, Ravi P; Hagmann, William K.
Afiliação
  • Li D; Departments of Medicinal Chemistry and Diabetes Research, Merck Research Laboratories , 126 East Lincoln Avenue, Rahway, New Jersey 07065, United States.
  • Wu Z; Departments of Medicinal Chemistry and Diabetes Research, Merck Research Laboratories , 126 East Lincoln Avenue, Rahway, New Jersey 07065, United States.
  • Yu Y; Departments of Medicinal Chemistry and Diabetes Research, Merck Research Laboratories , 126 East Lincoln Avenue, Rahway, New Jersey 07065, United States.
  • Ball RG; Departments of Medicinal Chemistry and Diabetes Research, Merck Research Laboratories , 126 East Lincoln Avenue, Rahway, New Jersey 07065, United States.
  • Guo L; Departments of Medicinal Chemistry and Diabetes Research, Merck Research Laboratories , 126 East Lincoln Avenue, Rahway, New Jersey 07065, United States.
  • Sherer E; Departments of Medicinal Chemistry and Diabetes Research, Merck Research Laboratories , 126 East Lincoln Avenue, Rahway, New Jersey 07065, United States.
  • He S; Departments of Medicinal Chemistry and Diabetes Research, Merck Research Laboratories , 126 East Lincoln Avenue, Rahway, New Jersey 07065, United States.
  • Hong Q; Departments of Medicinal Chemistry and Diabetes Research, Merck Research Laboratories , 126 East Lincoln Avenue, Rahway, New Jersey 07065, United States.
  • Lai Z; Departments of Medicinal Chemistry and Diabetes Research, Merck Research Laboratories , 126 East Lincoln Avenue, Rahway, New Jersey 07065, United States.
  • Qi H; Departments of Medicinal Chemistry and Diabetes Research, Merck Research Laboratories , 126 East Lincoln Avenue, Rahway, New Jersey 07065, United States.
  • Truong Q; Departments of Medicinal Chemistry and Diabetes Research, Merck Research Laboratories , 126 East Lincoln Avenue, Rahway, New Jersey 07065, United States.
  • Yang DX; Departments of Medicinal Chemistry and Diabetes Research, Merck Research Laboratories , 126 East Lincoln Avenue, Rahway, New Jersey 07065, United States.
  • Chicchi GG; Departments of Medicinal Chemistry and Diabetes Research, Merck Research Laboratories , 126 East Lincoln Avenue, Rahway, New Jersey 07065, United States.
  • Tsao KL; Departments of Medicinal Chemistry and Diabetes Research, Merck Research Laboratories , 126 East Lincoln Avenue, Rahway, New Jersey 07065, United States.
  • Trusca D; Departments of Medicinal Chemistry and Diabetes Research, Merck Research Laboratories , 126 East Lincoln Avenue, Rahway, New Jersey 07065, United States.
  • Trujillo M; Departments of Medicinal Chemistry and Diabetes Research, Merck Research Laboratories , 126 East Lincoln Avenue, Rahway, New Jersey 07065, United States.
  • Pachanski M; Departments of Medicinal Chemistry and Diabetes Research, Merck Research Laboratories , 126 East Lincoln Avenue, Rahway, New Jersey 07065, United States.
  • Eiermann GJ; Departments of Medicinal Chemistry and Diabetes Research, Merck Research Laboratories , 126 East Lincoln Avenue, Rahway, New Jersey 07065, United States.
  • Howard AD; Departments of Medicinal Chemistry and Diabetes Research, Merck Research Laboratories , 126 East Lincoln Avenue, Rahway, New Jersey 07065, United States.
  • Zhou YP; Departments of Medicinal Chemistry and Diabetes Research, Merck Research Laboratories , 126 East Lincoln Avenue, Rahway, New Jersey 07065, United States.
  • Zhang BB; Departments of Medicinal Chemistry and Diabetes Research, Merck Research Laboratories , 126 East Lincoln Avenue, Rahway, New Jersey 07065, United States.
  • Nargund RP; Departments of Medicinal Chemistry and Diabetes Research, Merck Research Laboratories , 126 East Lincoln Avenue, Rahway, New Jersey 07065, United States.
  • Hagmann WK; Departments of Medicinal Chemistry and Diabetes Research, Merck Research Laboratories , 126 East Lincoln Avenue, Rahway, New Jersey 07065, United States.
ACS Med Chem Lett ; 5(6): 690-5, 2014 Jun 12.
Article em En | MEDLINE | ID: mdl-24944745

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Idioma: En Revista: ACS Med Chem Lett Ano de publicação: 2014 Tipo de documento: Article País de afiliação: Estados Unidos

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Idioma: En Revista: ACS Med Chem Lett Ano de publicação: 2014 Tipo de documento: Article País de afiliação: Estados Unidos