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Solvent-Free Synthesis and Safener Activity of Sulfonylurea Benzothiazolines.
Fu, Ying; Wang, Jing-Yi; Zhang, Dong; Chen, Yu-Feng; Gao, Shuang; Zhao, Li-Xia; Ye, Fei.
Afiliação
  • Fu Y; Department of Applied Chemistry, College of Science, Northeast Agricultural University, Harbin 150030, China. fuying@neau.edu.cn.
  • Wang JY; Department of Applied Chemistry, College of Science, Northeast Agricultural University, Harbin 150030, China. wang-jingyi@foxmail.com.
  • Zhang D; Department of Applied Chemistry, College of Science, Northeast Agricultural University, Harbin 150030, China. zhangdong-qlc@163.com.
  • Chen YF; Department of Applied Chemistry, College of Science, Northeast Agricultural University, Harbin 150030, China. cyf1989919@163.com.
  • Gao S; Department of Applied Chemistry, College of Science, Northeast Agricultural University, Harbin 150030, China. gaoshuang@neau.edu.cn.
  • Zhao LX; Department of Applied Chemistry, College of Science, Northeast Agricultural University, Harbin 150030, China. zhaolixia@neau.edu.cn.
  • Ye F; Department of Applied Chemistry, College of Science, Northeast Agricultural University, Harbin 150030, China. yefei@neau.edu.cn.
Molecules ; 22(10)2017 Sep 22.
Article em En | MEDLINE | ID: mdl-28937640
ABSTRACT
A series of novel sulfonylurea benzothiazolines was designed by splicing active groups and bioisosterism. A solvent-free synthetic route was developed for the sulfonylurea benzothiazoline derivatives via the cyclization and carbamylation. All compounds were characterized by IR, ¹H-NMR, 13C-NMR, HRMS. The biological activity tests indicated the compounds could protect maize against the injury caused by chlorsulfuron to some extent. The molecular docking result showed that the new compound competed with chlorsulfuron to bind with the herbicide target enzyme active site to attain detoxification.
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Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Compostos de Sulfonilureia / Benzotiazóis Idioma: En Revista: Molecules Assunto da revista: BIOLOGIA Ano de publicação: 2017 Tipo de documento: Article País de afiliação: China
Texto completo
Imprimir
XML
PubMed Links
Buscar no Google

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Compostos de Sulfonilureia / Benzotiazóis Idioma: En Revista: Molecules Assunto da revista: BIOLOGIA Ano de publicação: 2017 Tipo de documento: Article País de afiliação: China