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Potent, selective, and subunit-dependent activation of TRPC5 channels by a xanthine derivative.
Minard, Aisling; Bauer, Claudia C; Chuntharpursat-Bon, Eulashini; Pickles, Isabelle B; Wright, David J; Ludlow, Melanie J; Burnham, Matthew P; Warriner, Stuart L; Beech, David J; Muraki, Katsuhiko; Bon, Robin S.
Afiliação
  • Minard A; School of Chemistry, University of Leeds, Leeds, UK.
  • Bauer CC; Department of Discovery and Translational Science, Leeds Institute of Cardiovascular and Metabolic Medicine, University of Leeds, Leeds, UK.
  • Chuntharpursat-Bon E; Department of Discovery and Translational Science, Leeds Institute of Cardiovascular and Metabolic Medicine, University of Leeds, Leeds, UK.
  • Pickles IB; Department of Discovery and Translational Science, Leeds Institute of Cardiovascular and Metabolic Medicine, University of Leeds, Leeds, UK.
  • Wright DJ; School of Chemistry, University of Leeds, Leeds, UK.
  • Ludlow MJ; Department of Discovery and Translational Science, Leeds Institute of Cardiovascular and Metabolic Medicine, University of Leeds, Leeds, UK.
  • Burnham MP; Department of Discovery and Translational Science, Leeds Institute of Cardiovascular and Metabolic Medicine, University of Leeds, Leeds, UK.
  • Warriner SL; Department of Discovery and Translational Science, Leeds Institute of Cardiovascular and Metabolic Medicine, University of Leeds, Leeds, UK.
  • Beech DJ; Discovery Sciences, R&B Biopharmaceuticals, AstraZeneca, Alderley Park, UK.
  • Muraki K; School of Chemistry, University of Leeds, Leeds, UK.
  • Bon RS; Department of Discovery and Translational Science, Leeds Institute of Cardiovascular and Metabolic Medicine, University of Leeds, Leeds, UK.
Br J Pharmacol ; 176(20): 3924-3938, 2019 10.
Article em En | MEDLINE | ID: mdl-31277085

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Purinas / Canais de Cátion TRPC / Compostos Heterocíclicos com 2 Anéis Limite: Humans Idioma: En Revista: Br J Pharmacol Ano de publicação: 2019 Tipo de documento: Article País de afiliação: Reino Unido

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Purinas / Canais de Cátion TRPC / Compostos Heterocíclicos com 2 Anéis Limite: Humans Idioma: En Revista: Br J Pharmacol Ano de publicação: 2019 Tipo de documento: Article País de afiliação: Reino Unido