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Discovery and antiviral profile of new sulfamoylbenzamide derivatives as HBV capsid assembly modulators.
Ivanova Bencheva, Leda; Donnici, Lorena; Ferrante, Luca; Prandi, Adolfo; Sinisi, Roberta; De Matteo, Marilenia; Randazzo, Pietro; Conti, Matteo; Di Lucia, Pietro; Bono, Elisa; Giustini, Leonardo; Vittoria Orsale, Maria; Patsilinakos, Alexandros; Monteagudo, Edith; Iannacone, Matteo; Summa, Vincenzo; Guidotti, Luca G; De Francesco, Raffaele; Di Fabio, Romano.
Afiliação
  • Ivanova Bencheva L; Promidis, Via Olgettina 60, 20132 Milano, Italy.
  • Donnici L; INGM, National Institute of Molecular Genetics "Romeo ed Enrica Invernizzi", Via Francesco Sforza, 35, 20122 Milan, Italy.
  • Ferrante L; Promidis, Via Olgettina 60, 20132 Milano, Italy.
  • Prandi A; Promidis, Via Olgettina 60, 20132 Milano, Italy.
  • Sinisi R; Promidis, Via Olgettina 60, 20132 Milano, Italy.
  • De Matteo M; Promidis, Via Olgettina 60, 20132 Milano, Italy.
  • Randazzo P; Promidis, Via Olgettina 60, 20132 Milano, Italy.
  • Conti M; INGM, National Institute of Molecular Genetics "Romeo ed Enrica Invernizzi", Via Francesco Sforza, 35, 20122 Milan, Italy.
  • Di Lucia P; Division of Immunology, Transplantation and Infectious Diseases, IRCCS San Raffaele Scientific Institute, Via Olgettina 60, 20132 Milan, Italy.
  • Bono E; Division of Immunology, Transplantation and Infectious Diseases, IRCCS San Raffaele Scientific Institute, Via Olgettina 60, 20132 Milan, Italy.
  • Giustini L; Division of Immunology, Transplantation and Infectious Diseases, IRCCS San Raffaele Scientific Institute, Via Olgettina 60, 20132 Milan, Italy.
  • Vittoria Orsale M; IRBM S.p.A., via Pontina Km 30.600, 00071 Pomezia (Rome), Italy.
  • Patsilinakos A; Sybilla Biotech S.r.l., via dei Solteri 38, 38131 Trento, Italy.
  • Monteagudo E; CHDI Foundation, 6080 Center Drive, Suite 700, Los Angeles, CA 90045, Italy.
  • Iannacone M; Division of Immunology, Transplantation and Infectious Diseases, IRCCS San Raffaele Scientific Institute, Via Olgettina 60, 20132 Milan, Italy; Vita-Salute San Raffaele University, Via Olgettina 60, 20132 Milan, Italy; Experimental Imaging Center, IRCCS San Raffaele Scientific Institute, Via Olgetti
  • Summa V; Department of Pharmacy, School of Medicine and Surgery, University of Naples Federico II, Vial Domenico Montesano 49, 80131 Naples, Italy.
  • Guidotti LG; Division of Immunology, Transplantation and Infectious Diseases, IRCCS San Raffaele Scientific Institute, Via Olgettina 60, 20132 Milan, Italy; Vita-Salute San Raffaele University, Via Olgettina 60, 20132 Milan, Italy.
  • De Francesco R; INGM, National Institute of Molecular Genetics "Romeo ed Enrica Invernizzi", Via Francesco Sforza, 35, 20122 Milan, Italy; Department of Pharmacological and Biomolecular Sciences, Università degli Studi di Milano, Via Balzaretti, 9, 20133 Milan, Italy.
  • Di Fabio R; Promidis, Via Olgettina 60, 20132 Milano, Italy; IRBM S.p.A., via Pontina Km 30.600, 00071 Pomezia (Rome), Italy. Electronic address: r.difabio@irbm.com.
Bioorg Med Chem Lett ; 73: 128904, 2022 10 01.
Article em En | MEDLINE | ID: mdl-35868496

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Antivirais / Capsídeo Limite: Animals Idioma: En Revista: Bioorg Med Chem Lett Assunto da revista: BIOQUIMICA / QUIMICA Ano de publicação: 2022 Tipo de documento: Article País de afiliação: Itália

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Antivirais / Capsídeo Limite: Animals Idioma: En Revista: Bioorg Med Chem Lett Assunto da revista: BIOQUIMICA / QUIMICA Ano de publicação: 2022 Tipo de documento: Article País de afiliação: Itália