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Identification of Histone Peptide Binding Specificity and Small-Molecule Ligands for the TRIM33α and TRIM33ß Bromodomains.
Sekirnik, Angelina R; Reynolds, Jessica K; See, Larissa; Bluck, Joseph P; Scorah, Amy R; Tallant, Cynthia; Lee, Bernadette; Leszczynska, Katarzyna B; Grimley, Rachel L; Storer, R Ian; Malattia, Marta; Crespillo, Sara; Caria, Sofia; Duclos, Stephanie; Hammond, Ester M; Knapp, Stefan; Morris, Garrett M; Duarte, Fernanda; Biggin, Philip C; Conway, Stuart J.
Afiliação
  • Sekirnik AR; Department of Chemistry, Chemistry Research Laboratory, University of Oxford, Mansfield Road, Oxford OX1 3TA, U.K.
  • Reynolds JK; Department of Chemistry, Chemistry Research Laboratory, University of Oxford, Mansfield Road, Oxford OX1 3TA, U.K.
  • See L; Department of Chemistry, Chemistry Research Laboratory, University of Oxford, Mansfield Road, Oxford OX1 3TA, U.K.
  • Bluck JP; Department of Chemistry, Chemistry Research Laboratory, University of Oxford, Mansfield Road, Oxford OX1 3TA, U.K.
  • Scorah AR; Department of Biochemistry, University of Oxford, South Parks Road, Oxford OX1 3QU, U.K.
  • Tallant C; Department of Chemistry, Chemistry Research Laboratory, University of Oxford, Mansfield Road, Oxford OX1 3TA, U.K.
  • Lee B; Nuffield Department of Clinical Medicine, Structural Genomics Consortium, University of Oxford, Old Road Campus Research Building, Roosevelt Drive, Oxford OX3 3TA, U.K.
  • Leszczynska KB; Department of Chemistry, Chemistry Research Laboratory, University of Oxford, Mansfield Road, Oxford OX1 3TA, U.K.
  • Grimley RL; Oxford Institute for Radiation Oncology, Department of Oncology, University of Oxford, Old Road Campus Research Building, Oxford OX3 7DQ, U.K.
  • Storer RI; Worldwide Medicinal Chemistry, Discovery Biology, Pfizer Ltd, The Portway, Granta Park, Cambridge CB21 6GS, U.K.
  • Malattia M; Worldwide Medicinal Chemistry, Discovery Biology, Pfizer Ltd, The Portway, Granta Park, Cambridge CB21 6GS, U.K.
  • Crespillo S; Evotec (UK) Ltd, 90 Park Drive, Milton Park, Abingdon, Oxfordshire OX14 4RZ, U.K.
  • Caria S; Evotec (UK) Ltd, 90 Park Drive, Milton Park, Abingdon, Oxfordshire OX14 4RZ, U.K.
  • Duclos S; Evotec (UK) Ltd, 90 Park Drive, Milton Park, Abingdon, Oxfordshire OX14 4RZ, U.K.
  • Hammond EM; Evotec (UK) Ltd, 90 Park Drive, Milton Park, Abingdon, Oxfordshire OX14 4RZ, U.K.
  • Knapp S; Oxford Institute for Radiation Oncology, Department of Oncology, University of Oxford, Old Road Campus Research Building, Oxford OX3 7DQ, U.K.
  • Morris GM; Institute of Pharmaceutical Chemistry, Goethe University, Max-von-Laue-Strasse 9, D-60438 Frankfurt am Main, Germany.
  • Duarte F; Structural Genomics Consortium, Buchmann Institute for Life Sciences (BMLS), Goethe University, Max-von-Laue-Strasse 15, D-60438 Frankfurt am Main, Germany.
  • Biggin PC; Department of Statistics, University of Oxford, 24-29 St Giles', Oxford OX1 3LB, U.K.
  • Conway SJ; Department of Chemistry, Chemistry Research Laboratory, University of Oxford, Mansfield Road, Oxford OX1 3TA, U.K.
ACS Chem Biol ; 17(10): 2753-2768, 2022 10 21.
Article em En | MEDLINE | ID: mdl-36098557

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Fatores de Transcrição / Histonas Tipo de estudo: Diagnostic_studies / Prognostic_studies Idioma: En Revista: ACS Chem Biol Ano de publicação: 2022 Tipo de documento: Article País de afiliação: Reino Unido

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Fatores de Transcrição / Histonas Tipo de estudo: Diagnostic_studies / Prognostic_studies Idioma: En Revista: ACS Chem Biol Ano de publicação: 2022 Tipo de documento: Article País de afiliação: Reino Unido