1.
Bioorg Med Chem Lett
; 19(1): 114-8, 2009 Jan 01.
Artículo
en Inglés
| MEDLINE
| ID: mdl-19014886
RESUMEN
A series of N-arylpiperazine camphor sulfonamides was discovered as novel CXCR3 antagonists. The synthesis, structure-activity relationships, and optimization of the initial hit that resulted in the identification of potent and selective CXCR3 antagonists are described.