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Bioorg Med Chem Lett
; 21(16): 4828-31, 2011 Aug 15.
Artículo
en Inglés
| MEDLINE
| ID: mdl-21741236
RESUMEN
Families of 2-arylbenzotriazoles and 2-arylindazoles that show positive effects in screens predictive of endogenous utrophin upregulation have been identified. Synthesis and structure-activity relationships are described leading to compounds with attractive in vitro profiles.