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Discovery of Brain-Penetrant, Irreversible Kynurenine Aminotransferase II Inhibitors for Schizophrenia.
Dounay, Amy B; Anderson, Marie; Bechle, Bruce M; Campbell, Brian M; Claffey, Michelle M; Evdokimov, Artem; Evrard, Edelweiss; Fonseca, Kari R; Gan, Xinmin; Ghosh, Somraj; Hayward, Matthew M; Horner, Weldon; Kim, Ji-Young; McAllister, Laura A; Pandit, Jayvardhan; Paradis, Vanessa; Parikh, Vinod D; Reese, Matthew R; Rong, SuoBao; Salafia, Michelle A; Schuyten, Katherine; Strick, Christine A; Tuttle, Jamison B; Valentine, James; Wang, Hong; Zawadzke, Laura E; Verhoest, Patrick R.
Afiliación
  • Dounay AB; Pfizer Worldwide Research and Development , Neuroscience Chemistry, Eastern Point Road, Groton, Connecticut 06340, United States.
  • Anderson M; Pfizer Worldwide Research and Development , Neuroscience Chemistry, Eastern Point Road, Groton, Connecticut 06340, United States.
  • Bechle BM; Pfizer Worldwide Research and Development , Neuroscience Chemistry, Eastern Point Road, Groton, Connecticut 06340, United States.
  • Campbell BM; Pfizer Worldwide Research and Development , Neuroscience Chemistry, Eastern Point Road, Groton, Connecticut 06340, United States.
  • Claffey MM; Pfizer Worldwide Research and Development , Neuroscience Chemistry, Eastern Point Road, Groton, Connecticut 06340, United States.
  • Evdokimov A; Pfizer Worldwide Research and Development , Neuroscience Chemistry, Eastern Point Road, Groton, Connecticut 06340, United States.
  • Evrard E; Pfizer Worldwide Research and Development , Neuroscience Chemistry, Eastern Point Road, Groton, Connecticut 06340, United States.
  • Fonseca KR; Pfizer Worldwide Research and Development , Neuroscience Chemistry, Eastern Point Road, Groton, Connecticut 06340, United States.
  • Gan X; Pfizer Worldwide Research and Development , Neuroscience Chemistry, Eastern Point Road, Groton, Connecticut 06340, United States.
  • Ghosh S; Pfizer Worldwide Research and Development , Neuroscience Chemistry, Eastern Point Road, Groton, Connecticut 06340, United States.
  • Hayward MM; Pfizer Worldwide Research and Development , Neuroscience Chemistry, Eastern Point Road, Groton, Connecticut 06340, United States.
  • Horner W; Pfizer Worldwide Research and Development , Neuroscience Chemistry, Eastern Point Road, Groton, Connecticut 06340, United States.
  • Kim JY; Pfizer Worldwide Research and Development , Neuroscience Chemistry, Eastern Point Road, Groton, Connecticut 06340, United States.
  • McAllister LA; Pfizer Worldwide Research and Development , Neuroscience Chemistry, Eastern Point Road, Groton, Connecticut 06340, United States.
  • Pandit J; Pfizer Worldwide Research and Development , Neuroscience Chemistry, Eastern Point Road, Groton, Connecticut 06340, United States.
  • Paradis V; Pfizer Worldwide Research and Development , Neuroscience Chemistry, Eastern Point Road, Groton, Connecticut 06340, United States.
  • Parikh VD; Pfizer Worldwide Research and Development , Neuroscience Chemistry, Eastern Point Road, Groton, Connecticut 06340, United States.
  • Reese MR; Pfizer Worldwide Research and Development , Neuroscience Chemistry, Eastern Point Road, Groton, Connecticut 06340, United States.
  • Rong S; Pfizer Worldwide Research and Development , Neuroscience Chemistry, Eastern Point Road, Groton, Connecticut 06340, United States.
  • Salafia MA; Pfizer Worldwide Research and Development , Neuroscience Chemistry, Eastern Point Road, Groton, Connecticut 06340, United States.
  • Schuyten K; Pfizer Worldwide Research and Development , Neuroscience Chemistry, Eastern Point Road, Groton, Connecticut 06340, United States.
  • Strick CA; Pfizer Worldwide Research and Development , Neuroscience Chemistry, Eastern Point Road, Groton, Connecticut 06340, United States.
  • Tuttle JB; Pfizer Worldwide Research and Development , Neuroscience Chemistry, Eastern Point Road, Groton, Connecticut 06340, United States.
  • Valentine J; Pfizer Worldwide Research and Development , Neuroscience Chemistry, Eastern Point Road, Groton, Connecticut 06340, United States.
  • Wang H; Pfizer Worldwide Research and Development , Neuroscience Chemistry, Eastern Point Road, Groton, Connecticut 06340, United States.
  • Zawadzke LE; Pfizer Worldwide Research and Development , Neuroscience Chemistry, Eastern Point Road, Groton, Connecticut 06340, United States.
  • Verhoest PR; Pfizer Worldwide Research and Development , Neuroscience Chemistry, Eastern Point Road, Groton, Connecticut 06340, United States.
ACS Med Chem Lett ; 3(3): 187-92, 2012 Mar 08.
Article en En | MEDLINE | ID: mdl-24900455

Texto completo: 1 Colección: 01-internacional Base de datos: MEDLINE Idioma: En Revista: ACS Med Chem Lett Año: 2012 Tipo del documento: Article País de afiliación: Estados Unidos

Texto completo: 1 Colección: 01-internacional Base de datos: MEDLINE Idioma: En Revista: ACS Med Chem Lett Año: 2012 Tipo del documento: Article País de afiliación: Estados Unidos
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