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Gaining in pan-affinity towards sigma 1 and sigma 2 receptors. SAR studies on arylalkylamines.
Rossi, Daniela; Rui, Marta; Di Giacomo, Marcello; Schepmann, Dirk; Wünsch, Bernhard; Monteleone, Stefania; Liedl, Klaus R; Collina, Simona.
Afiliación
  • Rossi D; Department of Drug Sciences, Medicinal Chemistry and Pharmaceutical Technology Section, University of Pavia, Viale Taramelli 12, 27100 Pavia, Italy.
  • Rui M; Department of Drug Sciences, Medicinal Chemistry and Pharmaceutical Technology Section, University of Pavia, Viale Taramelli 12, 27100 Pavia, Italy.
  • Di Giacomo M; Department of Drug Sciences, Medicinal Chemistry and Pharmaceutical Technology Section, University of Pavia, Viale Taramelli 12, 27100 Pavia, Italy.
  • Schepmann D; Institute of Pharmaceutical and Medicinal Chemistry, University of Muenster, Correnstrasse 48, 48149 Muenster, Germany.
  • Wünsch B; Institute of Pharmaceutical and Medicinal Chemistry, University of Muenster, Correnstrasse 48, 48149 Muenster, Germany.
  • Monteleone S; Institute of General, Inorganic and Theoretical Chemistry, Center of Molecular Biosciences, University of Innsbruck, Innrain 80/82, 6020 Innsbruck, Austria.
  • Liedl KR; Institute of General, Inorganic and Theoretical Chemistry, Center of Molecular Biosciences, University of Innsbruck, Innrain 80/82, 6020 Innsbruck, Austria.
  • Collina S; Department of Drug Sciences, Medicinal Chemistry and Pharmaceutical Technology Section, University of Pavia, Viale Taramelli 12, 27100 Pavia, Italy. Electronic address: simona.collina@unipv.it.
Bioorg Med Chem ; 25(1): 11-19, 2017 01 01.
Article en En | MEDLINE | ID: mdl-27838169

Texto completo: 1 Colección: 01-internacional Base de datos: MEDLINE Asunto principal: Receptores sigma / Descubrimiento de Drogas Tipo de estudio: Diagnostic_studies / Prognostic_studies Límite: Animals / Humans Idioma: En Revista: Bioorg Med Chem Asunto de la revista: BIOQUIMICA / QUIMICA Año: 2017 Tipo del documento: Article País de afiliación: Italia

Texto completo: 1 Colección: 01-internacional Base de datos: MEDLINE Asunto principal: Receptores sigma / Descubrimiento de Drogas Tipo de estudio: Diagnostic_studies / Prognostic_studies Límite: Animals / Humans Idioma: En Revista: Bioorg Med Chem Asunto de la revista: BIOQUIMICA / QUIMICA Año: 2017 Tipo del documento: Article País de afiliación: Italia
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