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Isoform-Selective ATAD2 Chemical Probe with Novel Chemical Structure and Unusual Mode of Action.
Fernández-Montalván, Amaury E; Berger, Markus; Kuropka, Benno; Koo, Seong Joo; Badock, Volker; Weiske, Joerg; Puetter, Vera; Holton, Simon J; Stöckigt, Detlef; Ter Laak, Antonius; Centrella, Paolo A; Clark, Matthew A; Dumelin, Christoph E; Sigel, Eric A; Soutter, Holly H; Troast, Dawn M; Zhang, Ying; Cuozzo, John W; Keefe, Anthony D; Roche, Didier; Rodeschini, Vincent; Chaikuad, Apirat; Díaz-Sáez, Laura; Bennett, James M; Fedorov, Oleg; Huber, Kilian V M; Hübner, Jan; Weinmann, Hilmar; Hartung, Ingo V; Gorjánácz, Mátyás.
Afiliación
  • Fernández-Montalván AE; Bayer AG , Pharmaceuticals, Drug Discovery, Berlin, Germany.
  • Berger M; Bayer AG , Pharmaceuticals, Drug Discovery, Berlin, Germany.
  • Kuropka B; Bayer AG , Pharmaceuticals, Drug Discovery, Berlin, Germany.
  • Koo SJ; Bayer AG , Pharmaceuticals, Drug Discovery, Berlin, Germany.
  • Badock V; Bayer AG , Pharmaceuticals, Drug Discovery, Berlin, Germany.
  • Weiske J; Bayer AG , Pharmaceuticals, Drug Discovery, Berlin, Germany.
  • Puetter V; Bayer AG , Pharmaceuticals, Drug Discovery, Berlin, Germany.
  • Holton SJ; Bayer AG , Pharmaceuticals, Drug Discovery, Berlin, Germany.
  • Stöckigt D; Bayer AG , Pharmaceuticals, Drug Discovery, Berlin, Germany.
  • Ter Laak A; Bayer AG , Pharmaceuticals, Drug Discovery, Berlin, Germany.
  • Centrella PA; X-Chem Pharmaceuticals , Waltham, Massachusetts United States.
  • Clark MA; X-Chem Pharmaceuticals , Waltham, Massachusetts United States.
  • Dumelin CE; X-Chem Pharmaceuticals , Waltham, Massachusetts United States.
  • Sigel EA; X-Chem Pharmaceuticals , Waltham, Massachusetts United States.
  • Soutter HH; X-Chem Pharmaceuticals , Waltham, Massachusetts United States.
  • Troast DM; X-Chem Pharmaceuticals , Waltham, Massachusetts United States.
  • Zhang Y; X-Chem Pharmaceuticals , Waltham, Massachusetts United States.
  • Cuozzo JW; X-Chem Pharmaceuticals , Waltham, Massachusetts United States.
  • Keefe AD; X-Chem Pharmaceuticals , Waltham, Massachusetts United States.
  • Roche D; Edelris , Lyon, France.
  • Rodeschini V; Edelris , Lyon, France.
  • Chaikuad A; Structural Genomics Consortium, Nuffield Department of Medicine, University of Oxford , Oxford, United Kingdom.
  • Díaz-Sáez L; Target Discovery Institute, Nuffield Department of Medicine, University of Oxford , Oxford, United Kingdom.
  • Bennett JM; Structural Genomics Consortium, Nuffield Department of Medicine, University of Oxford , Oxford, United Kingdom.
  • Fedorov O; Target Discovery Institute, Nuffield Department of Medicine, University of Oxford , Oxford, United Kingdom.
  • Huber KVM; Structural Genomics Consortium, Nuffield Department of Medicine, University of Oxford , Oxford, United Kingdom.
  • Hübner J; Target Discovery Institute, Nuffield Department of Medicine, University of Oxford , Oxford, United Kingdom.
  • Weinmann H; Structural Genomics Consortium, Nuffield Department of Medicine, University of Oxford , Oxford, United Kingdom.
  • Hartung IV; Target Discovery Institute, Nuffield Department of Medicine, University of Oxford , Oxford, United Kingdom.
  • Gorjánácz M; Structural Genomics Consortium, Nuffield Department of Medicine, University of Oxford , Oxford, United Kingdom.
ACS Chem Biol ; 12(11): 2730-2736, 2017 11 17.
Article en En | MEDLINE | ID: mdl-29043777

Texto completo: 1 Colección: 01-internacional Base de datos: MEDLINE Asunto principal: Sondas Moleculares / Proteínas de Unión al ADN / Multimerización de Proteína / Mapas de Interacción de Proteínas / ATPasas Asociadas con Actividades Celulares Diversas Límite: Humans Idioma: En Revista: ACS Chem Biol Año: 2017 Tipo del documento: Article País de afiliación: Alemania

Texto completo: 1 Colección: 01-internacional Base de datos: MEDLINE Asunto principal: Sondas Moleculares / Proteínas de Unión al ADN / Multimerización de Proteína / Mapas de Interacción de Proteínas / ATPasas Asociadas con Actividades Celulares Diversas Límite: Humans Idioma: En Revista: ACS Chem Biol Año: 2017 Tipo del documento: Article País de afiliación: Alemania
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