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Discovery of new potent molecular entities able to inhibit mPGES-1.
Di Micco, Simone; Terracciano, Stefania; Cantone, Vincenza; Fischer, Katrin; Koeberle, Andreas; Foglia, Antonio; Riccio, Raffaele; Werz, Oliver; Bruno, Ines; Bifulco, Giuseppe.
Afiliación
  • Di Micco S; Department of Pharmacy, University of Salerno, Via Giovanni Paolo II 132, 84084 Fisciano, Italy.
  • Terracciano S; Department of Pharmacy, University of Salerno, Via Giovanni Paolo II 132, 84084 Fisciano, Italy.
  • Cantone V; Department of Pharmacy, University of Salerno, Via Giovanni Paolo II 132, 84084 Fisciano, Italy; Department of Pharmaceutical/Medicinal Chemistry, Institute of Pharmacy, University of Jena, Philosophenweg 14, D-07743 Jena, Germany.
  • Fischer K; Department of Pharmaceutical/Medicinal Chemistry, Institute of Pharmacy, University of Jena, Philosophenweg 14, D-07743 Jena, Germany.
  • Koeberle A; Department of Pharmaceutical/Medicinal Chemistry, Institute of Pharmacy, University of Jena, Philosophenweg 14, D-07743 Jena, Germany.
  • Foglia A; Department of Pharmacy, University of Salerno, Via Giovanni Paolo II 132, 84084 Fisciano, Italy.
  • Riccio R; Department of Pharmacy, University of Salerno, Via Giovanni Paolo II 132, 84084 Fisciano, Italy.
  • Werz O; Department of Pharmaceutical/Medicinal Chemistry, Institute of Pharmacy, University of Jena, Philosophenweg 14, D-07743 Jena, Germany.
  • Bruno I; Department of Pharmacy, University of Salerno, Via Giovanni Paolo II 132, 84084 Fisciano, Italy. Electronic address: bruno@unisa.it.
  • Bifulco G; Department of Pharmacy, University of Salerno, Via Giovanni Paolo II 132, 84084 Fisciano, Italy. Electronic address: bifulco@unisa.it.
Eur J Med Chem ; 143: 1419-1427, 2018 Jan 01.
Article en En | MEDLINE | ID: mdl-29133047

Texto completo: 1 Colección: 01-internacional Base de datos: MEDLINE Asunto principal: Inhibidores Enzimáticos / Descubrimiento de Drogas / Prostaglandina-E Sintasas Tipo de estudio: Prognostic_studies Límite: Humans Idioma: En Revista: Eur J Med Chem Año: 2018 Tipo del documento: Article País de afiliación: Italia

Texto completo: 1 Colección: 01-internacional Base de datos: MEDLINE Asunto principal: Inhibidores Enzimáticos / Descubrimiento de Drogas / Prostaglandina-E Sintasas Tipo de estudio: Prognostic_studies Límite: Humans Idioma: En Revista: Eur J Med Chem Año: 2018 Tipo del documento: Article País de afiliación: Italia
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