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The Significance of Chirality in Drug Design and Synthesis of Bitopic Ligands as D3 Receptor (D3R) Selective Agonists.
Battiti, Francisco O; Cemaj, Sophie L; Guerrero, Adrian M; Shaik, Anver Basha; Lam, Jenny; Rais, Rana; Slusher, Barbara S; Deschamps, Jeffery R; Imler, Greg H; Newman, Amy Hauck; Bonifazi, Alessandro.
Afiliación
  • Battiti FO; Medicinal Chemistry Section, Molecular Targets and Medications Discovery Branch, National Institute on Drug Abuse-Intramural Research Program , National Institutes of Health , 333 Cassell Drive , Baltimore , Maryland 21224 , United States.
  • Cemaj SL; Medicinal Chemistry Section, Molecular Targets and Medications Discovery Branch, National Institute on Drug Abuse-Intramural Research Program , National Institutes of Health , 333 Cassell Drive , Baltimore , Maryland 21224 , United States.
  • Guerrero AM; Medicinal Chemistry Section, Molecular Targets and Medications Discovery Branch, National Institute on Drug Abuse-Intramural Research Program , National Institutes of Health , 333 Cassell Drive , Baltimore , Maryland 21224 , United States.
  • Shaik AB; Medicinal Chemistry Section, Molecular Targets and Medications Discovery Branch, National Institute on Drug Abuse-Intramural Research Program , National Institutes of Health , 333 Cassell Drive , Baltimore , Maryland 21224 , United States.
  • Lam J; Medicinal Chemistry Section, Molecular Targets and Medications Discovery Branch, National Institute on Drug Abuse-Intramural Research Program , National Institutes of Health , 333 Cassell Drive , Baltimore , Maryland 21224 , United States.
  • Rais R; Johns Hopkins Drug Discovery Program , Johns Hopkins School of Medicine , 855 N. Wolfe Street , Baltimore , Maryland 21205 , United States.
  • Slusher BS; Johns Hopkins Drug Discovery Program , Johns Hopkins School of Medicine , 855 N. Wolfe Street , Baltimore , Maryland 21205 , United States.
  • Deschamps JR; Johns Hopkins Drug Discovery Program , Johns Hopkins School of Medicine , 855 N. Wolfe Street , Baltimore , Maryland 21205 , United States.
  • Imler GH; Naval Research Laboratory , Code 6910, 4555 Overlook Avenue , Washington, DC 20375 , United States.
  • Newman AH; Naval Research Laboratory , Code 6910, 4555 Overlook Avenue , Washington, DC 20375 , United States.
  • Bonifazi A; Medicinal Chemistry Section, Molecular Targets and Medications Discovery Branch, National Institute on Drug Abuse-Intramural Research Program , National Institutes of Health , 333 Cassell Drive , Baltimore , Maryland 21224 , United States.
J Med Chem ; 62(13): 6287-6314, 2019 07 11.
Article en En | MEDLINE | ID: mdl-31257877

Texto completo: 1 Colección: 01-internacional Base de datos: MEDLINE Asunto principal: Agonistas de Dopamina / Receptores de Dopamina D3 / Indoles Límite: Animals / Humans Idioma: En Revista: J Med Chem Asunto de la revista: QUIMICA Año: 2019 Tipo del documento: Article País de afiliación: Estados Unidos

Texto completo: 1 Colección: 01-internacional Base de datos: MEDLINE Asunto principal: Agonistas de Dopamina / Receptores de Dopamina D3 / Indoles Límite: Animals / Humans Idioma: En Revista: J Med Chem Asunto de la revista: QUIMICA Año: 2019 Tipo del documento: Article País de afiliación: Estados Unidos
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