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Discovery of PqsE Thioesterase Inhibitors for Pseudomonas aeruginosa Using DNA-Encoded Small Molecule Library Screening.
Valastyan, Julie S; Tota, Michael R; Taylor, Isabelle R; Stergioula, Vasiliki; Hone, Graham A B; Smith, Chari D; Henke, Brad R; Carson, Kenneth G; Bassler, Bonnie L.
Afiliación
  • Valastyan JS; Department of Molecular Biology , Princeton University , Princeton , New Jersey 08544 , United States.
  • Tota MR; Howard Hughes Medical Institute , Chevy Chase , Maryland 20815 , United States.
  • Taylor IR; Macroceutics Incorporated, (now HotSpot Therapeutics) , Monmouth Junction , New Jersey 08852 , United States.
  • Stergioula V; Department of Molecular Biology , Princeton University , Princeton , New Jersey 08544 , United States.
  • Hone GAB; Department of Molecular Biology , Princeton University , Princeton , New Jersey 08544 , United States.
  • Smith CD; Macroceutics Incorporated, (now HotSpot Therapeutics) , Monmouth Junction , New Jersey 08852 , United States.
  • Henke BR; Department of Molecular Biology , Princeton University , Princeton , New Jersey 08544 , United States.
  • Carson KG; Opti-Mol Consulting, LLC , Cary , North Carolina 27513 , United States.
  • Bassler BL; Macroceutics Incorporated, (now HotSpot Therapeutics) , Monmouth Junction , New Jersey 08852 , United States.
ACS Chem Biol ; 15(2): 446-456, 2020 02 21.
Article en En | MEDLINE | ID: mdl-31880429

Texto completo: 1 Colección: 01-internacional Base de datos: MEDLINE Asunto principal: Pseudomonas aeruginosa / Tioléster Hidrolasas / Proteínas Bacterianas / ADN / Inhibidores Enzimáticos / Bibliotecas de Moléculas Pequeñas Tipo de estudio: Diagnostic_studies / Screening_studies Idioma: En Revista: ACS Chem Biol Año: 2020 Tipo del documento: Article País de afiliación: Estados Unidos

Texto completo: 1 Colección: 01-internacional Base de datos: MEDLINE Asunto principal: Pseudomonas aeruginosa / Tioléster Hidrolasas / Proteínas Bacterianas / ADN / Inhibidores Enzimáticos / Bibliotecas de Moléculas Pequeñas Tipo de estudio: Diagnostic_studies / Screening_studies Idioma: En Revista: ACS Chem Biol Año: 2020 Tipo del documento: Article País de afiliación: Estados Unidos
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