Lead Identification of 8-(Methylamino)-2-oxo-1,2-dihydroquinoline Derivatives as DNA Gyrase Inhibitors: Hit-to-Lead Generation Involving Thermodynamic Evaluation.

Ushiyama, Fumihito; Amada, Hideaki; Takeuchi, Tomoki; Tanaka-Yamamoto, Nozomi; Kanazawa, Harumi; Nakano, Koichiro; Mima, Masashi; Masuko, Aiko; Takata, Iichiro; Hitaka, Kosuke; Iwamoto, Kunihiko; Sugiyama, Hiroyuki; Ohtake, Norikazu

Ushiyama, Fumihito; Amada, Hideaki; Takeuchi, Tomoki; Tanaka-Yamamoto, Nozomi; Kanazawa, Harumi; Nakano, Koichiro; Mima, Masashi; Masuko, Aiko; Takata, Iichiro; Hitaka, Kosuke; Iwamoto, Kunihiko; Sugiyama, Hiroyuki; Ohtake, Norikazu.

Afiliación

Ushiyama F; Chemistry Laboratories, Taisho Pharmaceutical Company Ltd., 1-403, Yoshino-Cho, Kita-Ku, Saitama, Saitama 331-9530, Japan.
Amada H; Chemistry Laboratories, Taisho Pharmaceutical Company Ltd., 1-403, Yoshino-Cho, Kita-Ku, Saitama, Saitama 331-9530, Japan.
Takeuchi T; Chemistry Laboratories, Taisho Pharmaceutical Company Ltd., 1-403, Yoshino-Cho, Kita-Ku, Saitama, Saitama 331-9530, Japan.
Tanaka-Yamamoto N; Chemistry Laboratories, Taisho Pharmaceutical Company Ltd., 1-403, Yoshino-Cho, Kita-Ku, Saitama, Saitama 331-9530, Japan.
Kanazawa H; Chemistry Laboratories, Taisho Pharmaceutical Company Ltd., 1-403, Yoshino-Cho, Kita-Ku, Saitama, Saitama 331-9530, Japan.
Nakano K; Pharmacology Laboratories, Taisho Pharmaceutical Company Ltd., 1-403, Yoshino-Cho, Kita-Ku, Saitama, Saitama 331-9530, Japan.
Mima M; Pharmacology Laboratories, Taisho Pharmaceutical Company Ltd., 1-403, Yoshino-Cho, Kita-Ku, Saitama, Saitama 331-9530, Japan.
Masuko A; Pharmacology Laboratories, Taisho Pharmaceutical Company Ltd., 1-403, Yoshino-Cho, Kita-Ku, Saitama, Saitama 331-9530, Japan.
Takata I; Pharmacology Laboratories, Taisho Pharmaceutical Company Ltd., 1-403, Yoshino-Cho, Kita-Ku, Saitama, Saitama 331-9530, Japan.
Hitaka K; Pharmacology Laboratories, Taisho Pharmaceutical Company Ltd., 1-403, Yoshino-Cho, Kita-Ku, Saitama, Saitama 331-9530, Japan.
Iwamoto K; Pharmacology Laboratories, Taisho Pharmaceutical Company Ltd., 1-403, Yoshino-Cho, Kita-Ku, Saitama, Saitama 331-9530, Japan.
Sugiyama H; Pharmacology Laboratories, Taisho Pharmaceutical Company Ltd., 1-403, Yoshino-Cho, Kita-Ku, Saitama, Saitama 331-9530, Japan.
Ohtake N; Chemistry Laboratories, Taisho Pharmaceutical Company Ltd., 1-403, Yoshino-Cho, Kita-Ku, Saitama, Saitama 331-9530, Japan.

ACS Omega ; 5(17): 10145-10159, 2020 May 05.

Article en En | MEDLINE | ID: mdl-32391502

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Texto completo: 1 Colección: 01-internacional Base de datos: MEDLINE Tipo de estudio: Diagnostic_studies Idioma: En Revista: ACS Omega Año: 2020 Tipo del documento: Article País de afiliación: Japón

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