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Discovery and Structural Optimization of 4-(Aminomethyl)benzamides as Potent Entry Inhibitors of Ebola and Marburg Virus Infections.
Gaisina, Irina N; Peet, Norton P; Wong, Letitia; Schafer, Adam M; Cheng, Han; Anantpadma, Manu; Davey, Robert A; Thatcher, Gregory R J; Rong, Lijun.
Afiliación
  • Gaisina IN; UICentre (Drug Discovery @ UIC) and Department of Pharmaceutical Sciences, College of Pharmacy, University of Illinois at Chicago, 833 South Wood Street, Chicago, Illinois 60612, United States.
  • Peet NP; Chicago BioSolutions Inc., 2242 W Harrison Street, Chicago, Illinois 60612, United States.
  • Wong L; Chicago BioSolutions Inc., 2242 W Harrison Street, Chicago, Illinois 60612, United States.
  • Schafer AM; Chicago BioSolutions Inc., 2242 W Harrison Street, Chicago, Illinois 60612, United States.
  • Cheng H; College of Medicine, Department of Microbiology and Immunology, University of Illinois at Chicago, 909 S Wolcott Ave, Chicago, Illinois 60612, United States.
  • Anantpadma M; College of Medicine, Department of Microbiology and Immunology, University of Illinois at Chicago, 909 S Wolcott Ave, Chicago, Illinois 60612, United States.
  • Davey RA; Texas Biomedical Research Institute, 8715 W Military Drive, San Antonio, Texas 78227, United States.
  • Thatcher GRJ; Department of Microbiology, Boston University, 620 Albany Street, Boston, Massachusetts 02118, United States.
  • Rong L; Texas Biomedical Research Institute, 8715 W Military Drive, San Antonio, Texas 78227, United States.
J Med Chem ; 63(13): 7211-7225, 2020 07 09.
Article en En | MEDLINE | ID: mdl-32490678

Texto completo: 1 Colección: 01-internacional Base de datos: MEDLINE Asunto principal: Antivirales / Benzamidas / Fiebre Hemorrágica Ebola / Internalización del Virus / Enfermedad del Virus de Marburg Límite: Animals / Humans Idioma: En Revista: J Med Chem Asunto de la revista: QUIMICA Año: 2020 Tipo del documento: Article País de afiliación: Estados Unidos

Texto completo: 1 Colección: 01-internacional Base de datos: MEDLINE Asunto principal: Antivirales / Benzamidas / Fiebre Hemorrágica Ebola / Internalización del Virus / Enfermedad del Virus de Marburg Límite: Animals / Humans Idioma: En Revista: J Med Chem Asunto de la revista: QUIMICA Año: 2020 Tipo del documento: Article País de afiliación: Estados Unidos
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