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The novel potent TEAD inhibitor, K-975, inhibits YAP1/TAZ-TEAD protein-protein interactions and exerts an anti-tumor effect on malignant pleural mesothelioma.
Kaneda, Ayumi; Seike, Toshihiro; Danjo, Tomohiro; Nakajima, Takahiro; Otsubo, Nobumasa; Yamaguchi, Daisuke; Tsuji, Yoshiro; Hamaguchi, Kaori; Yasunaga, Mai; Nishiya, Yoichi; Suzuki, Michihiko; Saito, Jun-Ichi; Yatsunami, Rie; Nakamura, Satoshi; Sekido, Yoshitaka; Mori, Kiyotoshi.
Afiliación
  • Kaneda A; R&D Division, Kyowa Kirin Co., Ltd Shizuoka, Japan.
  • Seike T; School of Life Science and Technology, Tokyo Institute of Technology Yokohama, Japan.
  • Danjo T; R&D Division, Kyowa Kirin Co., Ltd Shizuoka, Japan.
  • Nakajima T; R&D Division, Kyowa Kirin Co., Ltd Shizuoka, Japan.
  • Otsubo N; R&D Division, Kyowa Kirin Co., Ltd Shizuoka, Japan.
  • Yamaguchi D; R&D Division, Kyowa Kirin Co., Ltd Shizuoka, Japan.
  • Tsuji Y; R&D Division, Kyowa Kirin Co., Ltd Shizuoka, Japan.
  • Hamaguchi K; R&D Division, Kyowa Kirin Co., Ltd Shizuoka, Japan.
  • Yasunaga M; R&D Division, Kyowa Kirin Co., Ltd Shizuoka, Japan.
  • Nishiya Y; R&D Division, Kyowa Kirin Co., Ltd Shizuoka, Japan.
  • Suzuki M; R&D Division, Kyowa Kirin Co., Ltd Shizuoka, Japan.
  • Saito JI; R&D Division, Kyowa Kirin Co., Ltd Shizuoka, Japan.
  • Yatsunami R; R&D Division, Kyowa Kirin Co., Ltd Shizuoka, Japan.
  • Nakamura S; School of Life Science and Technology, Tokyo Institute of Technology Yokohama, Japan.
  • Sekido Y; School of Life Science and Technology, Tokyo Institute of Technology Yokohama, Japan.
  • Mori K; National Institute of Technology, Numazu College Shizuoka, Japan.
Am J Cancer Res ; 10(12): 4399-4415, 2020.
Article en En | MEDLINE | ID: mdl-33415007

Texto completo: 1 Colección: 01-internacional Base de datos: MEDLINE Tipo de estudio: Prognostic_studies Idioma: En Revista: Am J Cancer Res Año: 2020 Tipo del documento: Article País de afiliación: Japón

Texto completo: 1 Colección: 01-internacional Base de datos: MEDLINE Tipo de estudio: Prognostic_studies Idioma: En Revista: Am J Cancer Res Año: 2020 Tipo del documento: Article País de afiliación: Japón
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