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Design and synthesis of 4-acetoxypentanamide derivatives of spliceostatin A and their biological evaluation towards prostate cancer treatment.
Hirabayashi, Satoru; Tsuyuguchi, Yuko; Li, Yue; Ohta, Noriko; Yoshikawa, Yusuke; Lin, Bangzhong; Fumimoto, Megumi; Nunomura, Kazuto; Suzuki, Takeyuki; Haruta, Junichi; Nimura, Keisuke; Arisawa, Mitsuhiro.
Afiliación
  • Hirabayashi S; Graduate School of Pharmaceutical Sciences, Osaka University, Yamada-oka 1-6, Suita, Osaka 565-0871, Japan.
  • Tsuyuguchi Y; Graduate School of Pharmaceutical Sciences, Osaka University, Yamada-oka 1-6, Suita, Osaka 565-0871, Japan.
  • Li Y; Division of Gene Therapy Science, Department of Genome Biology, Graduate School of Medicine, Osaka University, Yamada-oka 2-2, Suita, Osaka 565-0871, Japan.
  • Ohta N; Division of Gene Therapy Science, Department of Genome Biology, Graduate School of Medicine, Osaka University, Yamada-oka 2-2, Suita, Osaka 565-0871, Japan.
  • Yoshikawa Y; Graduate School of Pharmaceutical Sciences, Osaka University, Yamada-oka 1-6, Suita, Osaka 565-0871, Japan.
  • Lin B; Graduate School of Pharmaceutical Sciences, Osaka University, Yamada-oka 1-6, Suita, Osaka 565-0871, Japan.
  • Fumimoto M; Graduate School of Pharmaceutical Sciences, Osaka University, Yamada-oka 1-6, Suita, Osaka 565-0871, Japan.
  • Nunomura K; Graduate School of Pharmaceutical Sciences, Osaka University, Yamada-oka 1-6, Suita, Osaka 565-0871, Japan.
  • Suzuki T; Comprehensive Analysis Center, Sanken, Osaka University, Mihogaoka 8-1, Ibaraki, Osaka 567-0047, Japan.
  • Haruta J; Graduate School of Pharmaceutical Sciences, Osaka University, Yamada-oka 1-6, Suita, Osaka 565-0871, Japan.
  • Nimura K; Division of Gene Therapy Science, Department of Genome Biology, Graduate School of Medicine, Osaka University, Yamada-oka 2-2, Suita, Osaka 565-0871, Japan; Gunma University Initiative for Advanced Research, Gunma University, Showa-machi 3-39-22, Maebashi, Gunma 371-8511, Japan.
  • Arisawa M; Graduate School of Pharmaceutical Sciences, Osaka University, Yamada-oka 1-6, Suita, Osaka 565-0871, Japan. Electronic address: arisaw@phs.osaka-u.ac.jp.
Bioorg Med Chem Lett ; 91: 129333, 2023 07 15.
Article en En | MEDLINE | ID: mdl-37207846

Texto completo: 1 Colección: 01-internacional Base de datos: MEDLINE Asunto principal: Neoplasias de la Próstata / Compuestos de Espiro Límite: Humans / Male Idioma: En Revista: Bioorg Med Chem Lett Asunto de la revista: BIOQUIMICA / QUIMICA Año: 2023 Tipo del documento: Article País de afiliación: Japón

Texto completo: 1 Colección: 01-internacional Base de datos: MEDLINE Asunto principal: Neoplasias de la Próstata / Compuestos de Espiro Límite: Humans / Male Idioma: En Revista: Bioorg Med Chem Lett Asunto de la revista: BIOQUIMICA / QUIMICA Año: 2023 Tipo del documento: Article País de afiliación: Japón
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