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A potent and selective cis-amide inhibitor of ryanodine receptor 2 as a candidate for cardiac arrhythmia treatment.
Ishida, Ryosuke; Kurebayashi, Nagomi; Iinuma, Hiroto; Zeng, Xi; Mori, Shuichi; Kodama, Masami; Murayama, Takashi; Masuno, Hiroyuki; Takeda, Fumi; Kawahata, Masatoshi; Tanatani, Aya; Miura, Aya; Nishio, Hajime; Sakurai, Takashi; Kagechika, Hiroyuki.
Afiliación
  • Ishida R; Institute of Biomaterials and Bioengineering, Tokyo Medical and Dental University (TMDU), Tokyo, 101-0062, Japan.
  • Kurebayashi N; Department of Cellular and Molecular Pharmacology, Juntendo University Graduate School of Medicine, Tokyo, 113-8421, Japan. Electronic address: nagomik@juntendo.ac.jp.
  • Iinuma H; Institute of Biomaterials and Bioengineering, Tokyo Medical and Dental University (TMDU), Tokyo, 101-0062, Japan.
  • Zeng X; Institute of Biomaterials and Bioengineering, Tokyo Medical and Dental University (TMDU), Tokyo, 101-0062, Japan.
  • Mori S; Institute of Biomaterials and Bioengineering, Tokyo Medical and Dental University (TMDU), Tokyo, 101-0062, Japan.
  • Kodama M; Department of Cellular and Molecular Pharmacology, Juntendo University Graduate School of Medicine, Tokyo, 113-8421, Japan.
  • Murayama T; Department of Cellular and Molecular Pharmacology, Juntendo University Graduate School of Medicine, Tokyo, 113-8421, Japan.
  • Masuno H; Institute of Biomaterials and Bioengineering, Tokyo Medical and Dental University (TMDU), Tokyo, 101-0062, Japan.
  • Takeda F; Department of Chemistry, Faculty of Science, Ochanomizu University, 2-1-1 Otsuka, Bunkyo-ku, Tokyo, 112-8610, Japan.
  • Kawahata M; Faculty of Pharmaceutical Sciences, Showa Pharmaceutical University, 3-3165 Higashi-Tamagawagakuen, Machida, Tokyo, 194-8543, Japan.
  • Tanatani A; Department of Chemistry, Faculty of Science, Ochanomizu University, 2-1-1 Otsuka, Bunkyo-ku, Tokyo, 112-8610, Japan.
  • Miura A; Department of Legal Medicine, Hyogo Medical University, Nishinomiya, 663-8501, Japan.
  • Nishio H; Department of Legal Medicine, Hyogo Medical University, Nishinomiya, 663-8501, Japan.
  • Sakurai T; Department of Cellular and Molecular Pharmacology, Juntendo University Graduate School of Medicine, Tokyo, 113-8421, Japan.
  • Kagechika H; Institute of Biomaterials and Bioengineering, Tokyo Medical and Dental University (TMDU), Tokyo, 101-0062, Japan. Electronic address: kage.chem@tmd.ac.jp.
Eur J Med Chem ; 262: 115910, 2023 Dec 15.
Article en En | MEDLINE | ID: mdl-37922828

Texto completo: 1 Colección: 01-internacional Base de datos: MEDLINE Asunto principal: Canal Liberador de Calcio Receptor de Rianodina / Amidas Límite: Animals Idioma: En Revista: Eur J Med Chem Año: 2023 Tipo del documento: Article País de afiliación: Japón

Texto completo: 1 Colección: 01-internacional Base de datos: MEDLINE Asunto principal: Canal Liberador de Calcio Receptor de Rianodina / Amidas Límite: Animals Idioma: En Revista: Eur J Med Chem Año: 2023 Tipo del documento: Article País de afiliación: Japón
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