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Structural analogues of roscovitine rescue the intracellular traffic and the function of ER-retained ABCB4 variants in cell models.
Vauthier, Virginie; Ben Saad, Amel; Elie, Jonathan; Oumata, Nassima; Durand-Schneider, Anne-Marie; Bruneau, Alix; Delaunay, Jean-Louis; Housset, Chantal; Aït-Slimane, Tounsia; Meijer, Laurent; Falguières, Thomas.
Afiliação
  • Vauthier V; Inserm, Sorbonne Université, Centre de Recherche Saint-Antoine (CRSA), UMR_S 938, Institute of Cardiometabolism and Nutrition (ICAN), F-75012, Paris, France.
  • Ben Saad A; Inserm, Sorbonne Université, Centre de Recherche Saint-Antoine (CRSA), UMR_S 938, Institute of Cardiometabolism and Nutrition (ICAN), F-75012, Paris, France.
  • Elie J; ManRos Therapeutics, Hôtel de Recherche, Centre de Perharidy, F-29680, Roscoff, France.
  • Oumata N; ManRos Therapeutics, Hôtel de Recherche, Centre de Perharidy, F-29680, Roscoff, France.
  • Durand-Schneider AM; Inserm, Sorbonne Université, Centre de Recherche Saint-Antoine (CRSA), UMR_S 938, Institute of Cardiometabolism and Nutrition (ICAN), F-75012, Paris, France.
  • Bruneau A; Inserm, Sorbonne Université, Centre de Recherche Saint-Antoine (CRSA), UMR_S 938, Institute of Cardiometabolism and Nutrition (ICAN), F-75012, Paris, France.
  • Delaunay JL; Inserm, Sorbonne Université, Centre de Recherche Saint-Antoine (CRSA), UMR_S 938, Institute of Cardiometabolism and Nutrition (ICAN), F-75012, Paris, France.
  • Housset C; Inserm, Sorbonne Université, Centre de Recherche Saint-Antoine (CRSA), UMR_S 938, Institute of Cardiometabolism and Nutrition (ICAN), F-75012, Paris, France.
  • Aït-Slimane T; Assistance Publique - Hôpitaux de Paris, Hôpital Saint-Antoine, Centre de Référence des Maladies Rares - Maladies Inflammatoires des Voies Biliaires & Service d'Hépatologie, F-75012, Paris, France.
  • Meijer L; Inserm, Sorbonne Université, Centre de Recherche Saint-Antoine (CRSA), UMR_S 938, Institute of Cardiometabolism and Nutrition (ICAN), F-75012, Paris, France.
  • Falguières T; ManRos Therapeutics, Hôtel de Recherche, Centre de Perharidy, F-29680, Roscoff, France.
Sci Rep ; 9(1): 6653, 2019 04 30.
Article em En | MEDLINE | ID: mdl-31040306

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Subfamília B de Transportador de Cassetes de Ligação de ATP / Inibidores de Proteínas Quinases / Retículo Endoplasmático / Roscovitina / Antineoplásicos Limite: Humans Idioma: En Revista: Sci Rep Ano de publicação: 2019 Tipo de documento: Article País de afiliação: França

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Subfamília B de Transportador de Cassetes de Ligação de ATP / Inibidores de Proteínas Quinases / Retículo Endoplasmático / Roscovitina / Antineoplásicos Limite: Humans Idioma: En Revista: Sci Rep Ano de publicação: 2019 Tipo de documento: Article País de afiliação: França
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