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In Vivo Modulation of Cervicovaginal Drug Transporters and Tissue Distribution by Film-Released Tenofovir and Darunavir for Topical Prevention of HIV-1.
Hijazi, Karolin; Iannelli, Francesco; Cuppone, Anna Maria; Desjardins, Delphine; Caldwell, Anna; Dereuddre-Bosquet, Nathalie; Scala, Carlo; Smith, Kieron A; Mukhopadya, Indrani; Frank, Bruce; Gwozdz, Garry; Santoro, Francesco; Grand, Roger Le; Pozzi, Gianni; Kelly, Charles.
Afiliação
  • Hijazi K; Institute of Dentistry, School of Medicine Medical Sciences & Nutrition, University of Aberdeen, Aberdeen AB25 2ZR, U.K.
  • Iannelli F; Laboratory of Molecular Microbiology and Biotechnology, Department of Medical Biotechnologies, University of Siena, Siena 53100, Italy.
  • Cuppone AM; Laboratory of Molecular Microbiology and Biotechnology, Department of Medical Biotechnologies, University of Siena, Siena 53100, Italy.
  • Desjardins D; Université Paris Sud, INSERM U1184-Immunology of Viral Infections and Autoimmune Diseases (IMVA), IDMIT Department, IBFJ, CEA, Fontenay-aux-Roses, France.
  • Caldwell A; Mass Spectrometry Facility, King's College London, London SE1 9NH, U.K.
  • Dereuddre-Bosquet N; Université Paris Sud, INSERM U1184-Immunology of Viral Infections and Autoimmune Diseases (IMVA), IDMIT Department, IBFJ, CEA, Fontenay-aux-Roses, France.
  • Scala C; Faculty of Dentistry, Oral & Craniofacial Sciences, King's College London, London SE1 1UL, U.K.
  • Smith KA; Institute of Dentistry, School of Medicine Medical Sciences & Nutrition, University of Aberdeen, Aberdeen AB25 2ZR, U.K.
  • Mukhopadya I; Institute of Dentistry, School of Medicine Medical Sciences & Nutrition, University of Aberdeen, Aberdeen AB25 2ZR, U.K.
  • Frank B; Particle Sciences Inc., Lubrizol LifeSciences, Suite 180 Bethlehem, Pennsylvania 18017, United States.
  • Gwozdz G; Particle Sciences Inc., Lubrizol LifeSciences, Suite 180 Bethlehem, Pennsylvania 18017, United States.
  • Santoro F; Laboratory of Molecular Microbiology and Biotechnology, Department of Medical Biotechnologies, University of Siena, Siena 53100, Italy.
  • Grand RL; Université Paris Sud, INSERM U1184-Immunology of Viral Infections and Autoimmune Diseases (IMVA), IDMIT Department, IBFJ, CEA, Fontenay-aux-Roses, France.
  • Pozzi G; Laboratory of Molecular Microbiology and Biotechnology, Department of Medical Biotechnologies, University of Siena, Siena 53100, Italy.
  • Kelly C; Faculty of Dentistry, Oral & Craniofacial Sciences, King's College London, London SE1 1UL, U.K.
Mol Pharm ; 17(3): 852-864, 2020 03 02.
Article em En | MEDLINE | ID: mdl-32017579

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Contexto em Saúde: 1_ASSA2030 / 2_ODS3 Problema de saúde: 1_doencas_nao_transmissiveis / 2_enfermedades_transmissibles Assunto principal: Vagina / Infecções por HIV / Regulação para Cima / HIV-1 / Inibidores da Protease de HIV / Proteínas Associadas à Resistência a Múltiplos Medicamentos / Composição de Medicamentos / Darunavir / Tenofovir Limite: Animals / Female / Humans Idioma: En Revista: Mol Pharm Assunto da revista: BIOLOGIA MOLECULAR / FARMACIA / FARMACOLOGIA Ano de publicação: 2020 Tipo de documento: Article País de afiliação: Reino Unido

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Contexto em Saúde: 1_ASSA2030 / 2_ODS3 Problema de saúde: 1_doencas_nao_transmissiveis / 2_enfermedades_transmissibles Assunto principal: Vagina / Infecções por HIV / Regulação para Cima / HIV-1 / Inibidores da Protease de HIV / Proteínas Associadas à Resistência a Múltiplos Medicamentos / Composição de Medicamentos / Darunavir / Tenofovir Limite: Animals / Female / Humans Idioma: En Revista: Mol Pharm Assunto da revista: BIOLOGIA MOLECULAR / FARMACIA / FARMACOLOGIA Ano de publicação: 2020 Tipo de documento: Article País de afiliação: Reino Unido
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