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Synthesis and in vitro evaluation of novel spiroketopyrazoles as acetyl-CoA carboxylase inhibitors and potential antitumor agents.
Huang, Tonghui; Wu, Xin; Yan, Shirong; Liu, Tianya; Yin, Xiaoxing.
Afiliação
  • Huang T; Jiangsu Key Laboratory of New Drug Research and Clinical Pharmacy, Xuzhou Medical University, 221004, Xuzhou, Jiangsu, China; Xuzhou Medical University Science Park, 221000, Xuzhou, Jiangsu, People's Republic of China. Electronic address: tonghhuang@xzhmu.edu.cn.
  • Wu X; Jiangsu Key Laboratory of New Drug Research and Clinical Pharmacy, Xuzhou Medical University, 221004, Xuzhou, Jiangsu, China.
  • Yan S; Jiangsu Key Laboratory of New Drug Research and Clinical Pharmacy, Xuzhou Medical University, 221004, Xuzhou, Jiangsu, China.
  • Liu T; Department of Pharmacy, The Affiliated Hospital of Xuzhou Medical University, 221002, Xuzhou, Jiangsu, China.
  • Yin X; Jiangsu Key Laboratory of New Drug Research and Clinical Pharmacy, Xuzhou Medical University, 221004, Xuzhou, Jiangsu, China. Electronic address: yinxx@xzhmu.edu.cn.
Eur J Med Chem ; 212: 113036, 2021 Feb 15.
Article em En | MEDLINE | ID: mdl-33276990

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Acetil-CoA Carboxilase / Pirazóis / Compostos de Espiro / Inibidores Enzimáticos / Antineoplásicos Limite: Humans Idioma: En Revista: Eur J Med Chem Ano de publicação: 2021 Tipo de documento: Article

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Acetil-CoA Carboxilase / Pirazóis / Compostos de Espiro / Inibidores Enzimáticos / Antineoplásicos Limite: Humans Idioma: En Revista: Eur J Med Chem Ano de publicação: 2021 Tipo de documento: Article
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