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Design and synthesis of the first indole-based blockers of Panx-1 channel.
Crocetti, Letizia; Guerrini, Gabriella; Puglioli, Sara; Giovannoni, Maria Paola; Di Cesare Mannelli, Lorenzo; Lucarini, Elena; Ghelardini, Carla; Wang, Junjie; Dahl, Gerhard.
Afiliação
  • Crocetti L; Neurofarba, Pharmaceutical and Nutraceutical Section, University of Florence, Via Ugo Schiff 6, 50019, Sesto Fiorentino, Italy. Electronic address: letizia.crocetti@unifi.it.
  • Guerrini G; Neurofarba, Pharmaceutical and Nutraceutical Section, University of Florence, Via Ugo Schiff 6, 50019, Sesto Fiorentino, Italy. Electronic address: gabriella.guerrini@unifi.it.
  • Puglioli S; Neurofarba, Pharmaceutical and Nutraceutical Section, University of Florence, Via Ugo Schiff 6, 50019, Sesto Fiorentino, Italy. Electronic address: sara.puglioli@stud.unifi.it.
  • Giovannoni MP; Neurofarba, Pharmaceutical and Nutraceutical Section, University of Florence, Via Ugo Schiff 6, 50019, Sesto Fiorentino, Italy. Electronic address: mariapaola.giovannoni@unifi.it.
  • Di Cesare Mannelli L; Neurofarba, Pharmacology and Toxicology Section, University of Florence, Viale Pieraccini 6, 50139, Florence, Italy. Electronic address: lorenzo.mannelli@unifi.it.
  • Lucarini E; Neurofarba, Pharmacology and Toxicology Section, University of Florence, Viale Pieraccini 6, 50139, Florence, Italy. Electronic address: elena.lucarini@unifi.it.
  • Ghelardini C; Neurofarba, Pharmacology and Toxicology Section, University of Florence, Viale Pieraccini 6, 50139, Florence, Italy. Electronic address: carla.ghelardini@unifi.it.
  • Wang J; Department of Physiology and Biophysics, University of Miami School of Medicine, 1600 N.W. 10th Avenue Miami, Florida, 33136, USA. Electronic address: jwang1@miami.edu.
  • Dahl G; Department of Physiology and Biophysics, University of Miami School of Medicine, 1600 N.W. 10th Avenue Miami, Florida, 33136, USA. Electronic address: gdahl@miami.edu.
Eur J Med Chem ; 223: 113650, 2021 Nov 05.
Article em En | MEDLINE | ID: mdl-34174741

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Desenho de Fármacos / Indóis / Proteínas do Tecido Nervoso Limite: Animals / Humans / Male Idioma: En Revista: Eur J Med Chem Ano de publicação: 2021 Tipo de documento: Article

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Desenho de Fármacos / Indóis / Proteínas do Tecido Nervoso Limite: Animals / Humans / Male Idioma: En Revista: Eur J Med Chem Ano de publicação: 2021 Tipo de documento: Article
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