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Structure-based discovery of pyrazolamides as novel ERRγ inverse agonists.
Yang, Su Hui; Khadka, Daulat Bikram; Han, Jinhe; Na, Soon-Young; Shin, Minsang; Kim, Don-Kyu; Oh, Byung-Chul; Kim, Eun Young; Choi, Hueng-Sik; Cho, Won-Jea.
Afiliação
  • Yang SH; College of Pharmacy and Research Institute of Pharmaceutical Sciences, Chonnam National University, Gwang-ju, 61186, Republic of Korea.
  • Khadka DB; College of Pharmacy and Research Institute of Pharmaceutical Sciences, Chonnam National University, Gwang-ju, 61186, Republic of Korea.
  • Han J; College of Pharmacy and Research Institute of Pharmaceutical Sciences, Chonnam National University, Gwang-ju, 61186, Republic of Korea.
  • Na SY; School of Biological Sciences and Technology, Chonnam National University, Gwang-ju, 61186, Republic of Korea.
  • Shin M; Department of Microbiology, School of Medicine, Kyungpook National University, Deagu, 41944, Republic of Korea.
  • Kim DK; Department Integrative Food, Bioscience and Biotechnology, Chonnam National University, Gwang-ju, 61186, Republic of Korea.
  • Oh BC; Lee Gil Ya Cancer and Diabetes Institute, Gachon University Graduate School of Medicine, Incheon, 21564, Republic of Korea.
  • Kim EY; College of Pharmacy and Research Institute of Pharmaceutical Sciences, Chonnam National University, Gwang-ju, 61186, Republic of Korea.
  • Choi HS; School of Biological Sciences and Technology, Chonnam National University, Gwang-ju, 61186, Republic of Korea. Electronic address: hsc@jnu.ac.kr.
  • Cho WJ; College of Pharmacy and Research Institute of Pharmaceutical Sciences, Chonnam National University, Gwang-ju, 61186, Republic of Korea. Electronic address: wjcho@jnu.ac.kr.
Eur J Med Chem ; 250: 115174, 2023 Mar 15.
Article em En | MEDLINE | ID: mdl-36805944

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Receptores de Estrogênio / Agonismo Inverso de Drogas Idioma: En Revista: Eur J Med Chem Ano de publicação: 2023 Tipo de documento: Article

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Receptores de Estrogênio / Agonismo Inverso de Drogas Idioma: En Revista: Eur J Med Chem Ano de publicação: 2023 Tipo de documento: Article
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