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Discovery and Structure-Based Design of Inhibitors of the WD Repeat-Containing Protein 5 (WDR5)-MYC Interaction.
Ding, Jian; Liu, Lulu; Chiang, Ying-Ling; Zhao, Mengxi; Liu, Hejun; Yang, Fei; Shen, Lingling; Lin, Ying; Deng, Huiwen; Gao, Jingyan; Sage, David R; West, Laura; Llamas, Luis A; Hao, Xin; Kawatkar, Sameer; Li, En; Jain, Rishi K; Tallarico, John A; Canham, Stephen M; Wang, He.
Afiliação
  • Ding J; Novartis Institutes for BioMedical Research, Cambridge, Massachusetts 02139, United States.
  • Liu L; Novartis Institutes for BioMedical Research, Cambridge, Massachusetts 02139, United States.
  • Chiang YL; Novartis Institutes for BioMedical Research, Cambridge, Massachusetts 02139, United States.
  • Zhao M; Novartis Institutes for BioMedical Research, Shanghai 201203, China.
  • Liu H; Novartis Institutes for BioMedical Research, Shanghai 201203, China.
  • Yang F; Novartis Institutes for BioMedical Research, Shanghai 201203, China.
  • Shen L; Novartis Institutes for BioMedical Research, San Diego, California 92121, United States.
  • Lin Y; Novartis Institutes for BioMedical Research, Cambridge, Massachusetts 02139, United States.
  • Deng H; Novartis Institutes for BioMedical Research, Cambridge, Massachusetts 02139, United States.
  • Gao J; Novartis Institutes for BioMedical Research, Shanghai 201203, China.
  • Sage DR; Novartis Institutes for BioMedical Research, Shanghai 201203, China.
  • West L; Novartis Institutes for BioMedical Research, Shanghai 201203, China.
  • Llamas LA; Novartis Institutes for BioMedical Research, Cambridge, Massachusetts 02139, United States.
  • Hao X; Novartis Institutes for BioMedical Research, Cambridge, Massachusetts 02139, United States.
  • Kawatkar S; Novartis Institutes for BioMedical Research, Cambridge, Massachusetts 02139, United States.
  • Li E; Novartis Institutes for BioMedical Research, Shanghai 201203, China.
  • Jain RK; Novartis Institutes for BioMedical Research, Cambridge, Massachusetts 02139, United States.
  • Tallarico JA; Novartis Institutes for BioMedical Research, Shanghai 201203, China.
  • Canham SM; Novartis Institutes for BioMedical Research, Cambridge, Massachusetts 02139, United States.
  • Wang H; Novartis Institutes for BioMedical Research, Cambridge, Massachusetts 02139, United States.
J Med Chem ; 66(12): 8310-8323, 2023 06 22.
Article em En | MEDLINE | ID: mdl-37307526

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Repetições WD40 / Neoplasias Limite: Humans Idioma: En Revista: J Med Chem Assunto da revista: QUIMICA Ano de publicação: 2023 Tipo de documento: Article País de afiliação: Estados Unidos

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Repetições WD40 / Neoplasias Limite: Humans Idioma: En Revista: J Med Chem Assunto da revista: QUIMICA Ano de publicação: 2023 Tipo de documento: Article País de afiliação: Estados Unidos
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