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X-Ray Conformation and Structure-Activity Relationships of MA026, a Reversible Tight Junction Opener.
Mukaiyama, Minagi; Uchiyama, Chihiro; Fukuda, Akane; Nakazawa, Yoshiki; Kuramochi, Yuka; Shibata, Yudai; Konno, Sho; Muguruma, Kyohei; Matsugaki, Naohiro; Asari, Tomo; Ogawa, Kazuyoshi; Taguchi, Akihiro; Takayama, Kentaro; Taniguchi, Atsuhiko; Nagumo, Yoko; Senda, Toshiya; Hayashi, Yoshio; Usui, Takeo.
Afiliação
  • Mukaiyama M; Graduate School of Science and Technology, University of Tsukuba, Tsukuba, Ibaraki 305-8572, Japan.
  • Uchiyama C; School of Pharmacy, Tokyo University of Pharmacy and Life Sciences, Hachioji, Tokyo 192-0392, Japan.
  • Fukuda A; School of Pharmacy, Tokyo University of Pharmacy and Life Sciences, Hachioji, Tokyo 192-0392, Japan.
  • Nakazawa Y; School of Pharmacy, Tokyo University of Pharmacy and Life Sciences, Hachioji, Tokyo 192-0392, Japan.
  • Kuramochi Y; School of Pharmacy, Tokyo University of Pharmacy and Life Sciences, Hachioji, Tokyo 192-0392, Japan.
  • Shibata Y; School of Pharmacy, Tokyo University of Pharmacy and Life Sciences, Hachioji, Tokyo 192-0392, Japan.
  • Konno S; School of Pharmacy, Tokyo University of Pharmacy and Life Sciences, Hachioji, Tokyo 192-0392, Japan.
  • Muguruma K; School of Pharmacy, Tokyo University of Pharmacy and Life Sciences, Hachioji, Tokyo 192-0392, Japan.
  • Matsugaki N; Structural Biology Research Center, High Energy Accelerator Research Organization (KEK), Institute of Materials Structure Science, Tsukuba, Ibaraki 305-0801, Japan.
  • Asari T; Department of Materials Structure Science, School of High Energy Accelerator Science, The Graduate University of Advanced Studies (Soken-dai), 1-1 Oho, Tsukuba, Tsukuba, Ibaraki 305-0801, Japan.
  • Ogawa K; School of Pharmacy, Tokyo University of Pharmacy and Life Sciences, Hachioji, Tokyo 192-0392, Japan.
  • Taguchi A; Alliance for Research on the Mediterranean and North Africa (ARENA), University of Tsukuba, Tsukuba, Ibaraki 305-8572, Japan.
  • Takayama K; School of Pharmacy, Tokyo University of Pharmacy and Life Sciences, Hachioji, Tokyo 192-0392, Japan.
  • Taniguchi A; School of Pharmacy, Tokyo University of Pharmacy and Life Sciences, Hachioji, Tokyo 192-0392, Japan.
  • Nagumo Y; School of Pharmacy, Tokyo University of Pharmacy and Life Sciences, Hachioji, Tokyo 192-0392, Japan.
  • Senda T; Alliance for Research on the Mediterranean and North Africa (ARENA), University of Tsukuba, Tsukuba, Ibaraki 305-8572, Japan.
  • Hayashi Y; Institute of Environmental Sciences, University of Tsukuba, Tsukuba, Ibaraki 305-8572, Japan.
  • Usui T; Institute of Pure and Applied Sciences, University of Tsukuba, Tsukuba, Ibaraki 305-8572, Japan.
J Med Chem ; 66(13): 8717-8724, 2023 07 13.
Article em En | MEDLINE | ID: mdl-37352439

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Junções Íntimas Idioma: En Revista: J Med Chem Assunto da revista: QUIMICA Ano de publicação: 2023 Tipo de documento: Article País de afiliação: Japão

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Junções Íntimas Idioma: En Revista: J Med Chem Assunto da revista: QUIMICA Ano de publicação: 2023 Tipo de documento: Article País de afiliação: Japão
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