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Parasitol Int ; 66(2): 47-55, 2017 Apr.
Artigo em Inglês | MEDLINE | ID: mdl-27888011

RESUMO

Leishmania (Leishmania) infantum chagasi is one of the agents that cause visceral leishmaniasis. This disease occurs more frequently in third world countries, such as Brazil. The treatment is arduous, and is dependent on just a few drugs like the antimonial derivatives and amphotericin B. Moreover, these drugs are not only expensive, but they can also cause severe side effects and require long-term treatment. Therefore, it is very important to find new compounds that are effective against leishmaniasis. In the present work we evaluated a new group of synthetic amides against the promastigote and amastigote forms of L. infantum chagasi. The results showed that one of these amides in particular, presented very effective activity against the promastigotes and amastigotes of L. infantum chagasi at low concentrations and it also presented low toxicity for mammal cells, which makes this synthetic amide a promising drug for combating leishmaniasis.


Assuntos
Antiprotozoários/farmacologia , Leishmania infantum/efeitos dos fármacos , Fenetilaminas/farmacologia , Animais , Antiprotozoários/síntese química , Antiprotozoários/química , Brasil , Linhagem Celular , Descoberta de Drogas , Leishmania/efeitos dos fármacos , Leishmania/ultraestrutura , Leishmania infantum/crescimento & desenvolvimento , Leishmania infantum/fisiologia , Leishmania infantum/ultraestrutura , Estágios do Ciclo de Vida/efeitos dos fármacos , Macrófagos Peritoneais/efeitos dos fármacos , Camundongos , Fenetilaminas/síntese química , Fenetilaminas/química
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