1.
Bioorg Med Chem Lett
; 18(15): 4428-32, 2008 Aug 01.
Artigo
em Inglês
| MEDLINE
| ID: mdl-18614366
RESUMO
The biphenyl amides (BPAs) are a novel series of p38alpha MAP kinase inhibitor. The optimisation of the series to give compounds that are potent in an in vivo disease model is discussed. SAR is presented and rationalised with reference to the crystallographic binding mode.