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Novel TKI-resistant BCR-ABL1 gatekeeper residue mutations retain in vitro sensitivity to axitinib.
Lasater, E A; Massi, E S; Stecula, A; Politi, J; Tan, S K; Smith, C C; Gunthorpe, M; Holmes, J P; Chehab, F; Sali, A; Shah, N P.
Affiliation
  • Lasater EA; Division of Hematology/Oncology, University of California, San Francisco, CA, USA.
  • Massi ES; Division of Hematology/Oncology, University of California, San Francisco, CA, USA.
  • Stecula A; Department of Bioengineering and Therapeutic Sciences, University of California, San Francisco, CA, USA.
  • Politi J; Division of Hematology/Oncology, University of California, San Francisco, CA, USA.
  • Tan SK; Division of Hematology/Oncology, University of California, San Francisco, CA, USA.
  • Smith CC; Division of Hematology/Oncology, University of California, San Francisco, CA, USA.
  • Gunthorpe M; Department of Laboratory Medicine, University of California, San Francisco, CA, USA.
  • Holmes JP; Annadel Medical Group, Santa Rosa, CA, USA.
  • Chehab F; Department of Laboratory Medicine, University of California, San Francisco, CA, USA.
  • Sali A; Department of Bioengineering and Therapeutic Sciences, University of California, San Francisco, CA, USA.
  • Shah NP; Department of Pharmaceutical Chemistry, University of California, San Francisco, CA, USA.
Leukemia ; 30(6): 1405-9, 2016 06.
Article in En | MEDLINE | ID: mdl-26511402

Full text: 1 Collection: 01-internacional Database: MEDLINE Main subject: Protein-Tyrosine Kinases / Fusion Proteins, bcr-abl / Protein Kinase Inhibitors / Imidazoles / Indazoles Type of study: Diagnostic_studies Limits: Humans / Male / Middle aged Language: En Journal: Leukemia Year: 2016 Document type: Article

Full text: 1 Collection: 01-internacional Database: MEDLINE Main subject: Protein-Tyrosine Kinases / Fusion Proteins, bcr-abl / Protein Kinase Inhibitors / Imidazoles / Indazoles Type of study: Diagnostic_studies Limits: Humans / Male / Middle aged Language: En Journal: Leukemia Year: 2016 Document type: Article