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Synthesis, Pharmacological Evaluation, and Docking Studies of Novel Pyridazinone-Based Cannabinoid Receptor Type 2 Ligands.
Ragusa, Giulio; Bencivenni, Serena; Morales, Paula; Callaway, Tyra; Hurst, Dow P; Asproni, Battistina; Merighi, Stefania; Loriga, Giovanni; Pinna, Gerard A; Reggio, Patricia H; Gessi, Stefania; Murineddu, Gabriele.
Affiliation
  • Ragusa G; Department of Chemistry and Pharmacy, University of Sassari, via F. Muroni 23/A, 07100, Sassari, Italy.
  • Bencivenni S; Dipartimento di Scienze Mediche, Sezione di Farmacologia, Università di Ferrara, Via Fossato di Mortara, 17-19, 44121, Ferrara, Italy.
  • Morales P; Department of Chemistry and Biochemistry, University of North Carolina at Greensboro, Greensboro, NC, 27402, USA.
  • Callaway T; Department of Chemistry and Biochemistry, University of North Carolina at Greensboro, Greensboro, NC, 27402, USA.
  • Hurst DP; Department of Chemistry and Biochemistry, University of North Carolina at Greensboro, Greensboro, NC, 27402, USA.
  • Asproni B; Department of Chemistry and Pharmacy, University of Sassari, via F. Muroni 23/A, 07100, Sassari, Italy.
  • Merighi S; Dipartimento di Scienze Mediche, Sezione di Farmacologia, Università di Ferrara, Via Fossato di Mortara, 17-19, 44121, Ferrara, Italy.
  • Loriga G; Institute of Translational Pharmacology, National Research Council, 09010 Pula, Cagliari, Italy.
  • Pinna GA; Department of Chemistry and Pharmacy, University of Sassari, via F. Muroni 23/A, 07100, Sassari, Italy.
  • Reggio PH; Department of Chemistry and Biochemistry, University of North Carolina at Greensboro, Greensboro, NC, 27402, USA.
  • Gessi S; Dipartimento di Scienze Mediche, Sezione di Farmacologia, Università di Ferrara, Via Fossato di Mortara, 17-19, 44121, Ferrara, Italy.
  • Murineddu G; Department of Chemistry and Pharmacy, University of Sassari, via F. Muroni 23/A, 07100, Sassari, Italy.
ChemMedChem ; 13(11): 1102-1114, 2018 06 06.
Article in En | MEDLINE | ID: mdl-29575721

Full text: 1 Collection: 01-internacional Database: MEDLINE Main subject: Pyridazines / Receptor, Cannabinoid, CB2 / Cannabinoid Receptor Antagonists Limits: Animals / Humans Language: En Journal: ChemMedChem Year: 2018 Document type: Article

Full text: 1 Collection: 01-internacional Database: MEDLINE Main subject: Pyridazines / Receptor, Cannabinoid, CB2 / Cannabinoid Receptor Antagonists Limits: Animals / Humans Language: En Journal: ChemMedChem Year: 2018 Document type: Article