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Synthesis and evaluation of 4-cycloheptylphenols as selective Estrogen receptor-ß agonists (SERBAs).
Sampathi Perera, K L Iresha; Hanson, Alicia M; Lindeman, Sergey; Imhoff, Andrea; Lu, Xingyun; Sem, Daniel S; Donaldson, William A.
Affiliation
  • Sampathi Perera KLI; Department of Chemistry, Marquette University, P. O. Box 1881, Milwaukee, WI, 53201-1881, United States.
  • Hanson AM; School of Pharmacy, Center for Structure-based Drug Design and Development, Concordia University Wisconsin, Mequon, WI, 53097, United States.
  • Lindeman S; Department of Chemistry, Marquette University, P. O. Box 1881, Milwaukee, WI, 53201-1881, United States.
  • Imhoff A; School of Pharmacy, Center for Structure-based Drug Design and Development, Concordia University Wisconsin, Mequon, WI, 53097, United States.
  • Lu X; School of Pharmacy, Center for Structure-based Drug Design and Development, Concordia University Wisconsin, Mequon, WI, 53097, United States.
  • Sem DS; School of Pharmacy, Center for Structure-based Drug Design and Development, Concordia University Wisconsin, Mequon, WI, 53097, United States.
  • Donaldson WA; Department of Chemistry, Marquette University, P. O. Box 1881, Milwaukee, WI, 53201-1881, United States. Electronic address: william.donaldson@marquette.edu.
Eur J Med Chem ; 157: 791-804, 2018 Sep 05.
Article in En | MEDLINE | ID: mdl-30144697

Full text: 1 Collection: 01-internacional Database: MEDLINE Main subject: Phenols / Cycloheptanes / Estrogen Receptor beta / Methanol / Estrogens / Antineoplastic Agents Limits: Humans Language: En Journal: Eur J Med Chem Year: 2018 Document type: Article

Full text: 1 Collection: 01-internacional Database: MEDLINE Main subject: Phenols / Cycloheptanes / Estrogen Receptor beta / Methanol / Estrogens / Antineoplastic Agents Limits: Humans Language: En Journal: Eur J Med Chem Year: 2018 Document type: Article