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Lenacapavir: A Novel, Potent, and Selective First-in-Class Inhibitor of HIV-1 Capsid Function Exhibits Optimal Pharmacokinetic Properties for a Long-Acting Injectable Antiretroviral Agent.
Subramanian, Raju; Tang, Jennifer; Zheng, Jim; Lu, Bing; Wang, Kelly; Yant, Stephen R; Stepan, George J; Mulato, Andrew; Yu, Helen; Schroeder, Scott; Shaik, Naveed; Singh, Renu; Wolckenhauer, Scott; Chester, Anne; Tse, Winston C; Chiu, Anna; Rhee, Martin; Cihlar, Tomas; Rowe, William; Smith, Bill J.
Affiliation
  • Subramanian R; Gilead Sciences, Inc., 333 Lakeside Drive, Foster City, California 94404, United States.
  • Tang J; Gilead Sciences, Inc., 333 Lakeside Drive, Foster City, California 94404, United States.
  • Zheng J; Gilead Sciences, Inc., 333 Lakeside Drive, Foster City, California 94404, United States.
  • Lu B; Gilead Sciences, Inc., 333 Lakeside Drive, Foster City, California 94404, United States.
  • Wang K; Gilead Sciences, Inc., 333 Lakeside Drive, Foster City, California 94404, United States.
  • Yant SR; Gilead Sciences, Inc., 333 Lakeside Drive, Foster City, California 94404, United States.
  • Stepan GJ; Gilead Sciences, Inc., 333 Lakeside Drive, Foster City, California 94404, United States.
  • Mulato A; Gilead Sciences, Inc., 333 Lakeside Drive, Foster City, California 94404, United States.
  • Yu H; Gilead Sciences, Inc., 333 Lakeside Drive, Foster City, California 94404, United States.
  • Schroeder S; Gilead Sciences, Inc., 333 Lakeside Drive, Foster City, California 94404, United States.
  • Shaik N; Gilead Sciences, Inc., 333 Lakeside Drive, Foster City, California 94404, United States.
  • Singh R; Gilead Sciences, Inc., 333 Lakeside Drive, Foster City, California 94404, United States.
  • Wolckenhauer S; Gilead Sciences, Inc., 333 Lakeside Drive, Foster City, California 94404, United States.
  • Chester A; Gilead Sciences, Inc., 333 Lakeside Drive, Foster City, California 94404, United States.
  • Tse WC; Gilead Sciences, Inc., 333 Lakeside Drive, Foster City, California 94404, United States.
  • Chiu A; Gilead Sciences, Inc., 333 Lakeside Drive, Foster City, California 94404, United States.
  • Rhee M; Gilead Sciences, Inc., 333 Lakeside Drive, Foster City, California 94404, United States.
  • Cihlar T; Gilead Sciences, Inc., 333 Lakeside Drive, Foster City, California 94404, United States.
  • Rowe W; Gilead Sciences, Inc., 333 Lakeside Drive, Foster City, California 94404, United States.
  • Smith BJ; Gilead Sciences, Inc., 333 Lakeside Drive, Foster City, California 94404, United States.
Mol Pharm ; 20(12): 6213-6225, 2023 Dec 04.
Article in En | MEDLINE | ID: mdl-37917742

Full text: 1 Collection: 01-internacional Database: MEDLINE Main subject: HIV-1 / Anti-HIV Agents Limits: Animals / Humans Language: En Journal: Mol Pharm Year: 2023 Document type: Article

Full text: 1 Collection: 01-internacional Database: MEDLINE Main subject: HIV-1 / Anti-HIV Agents Limits: Animals / Humans Language: En Journal: Mol Pharm Year: 2023 Document type: Article