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Identification of a selective inhibitor of murine intestinal alkaline phosphatase (ML260) by concurrent ultra-high throughput screening against human and mouse isozymes.
Ardecky, Robert J; Bobkova, Ekaterina V; Kiffer-Moreira, Tina; Brown, Brock; Ganji, Santhi; Zou, Jiwen; Pass, Ian; Narisawa, Sonoko; Iano, Flávia Godoy; Rosenstein, Craig; Cheltsov, Anton; Rascon, Justin; Hedrick, Michael; Gasior, Carlton; Forster, Anita; Shi, Shenghua; Dahl, Russell; Vasile, Stefan; Su, Ying; Sergienko, Eduard; Chung, Thomas D Y; Kaunitz, Jonathan; Hoylaerts, Marc F; Pinkerton, Anthony B; Millán, José Luis.
Afiliação
  • Ardecky RJ; Sanford-Burnham Medical Research Institute, La Jolla, CA 92037.
  • Bobkova EV; Sanford-Burnham Medical Research Institute, La Jolla, CA 92037.
  • Kiffer-Moreira T; Sanford-Burnham Medical Research Institute, La Jolla, CA 92037.
  • Brown B; Sanford-Burnham Medical Research Institute, La Jolla, CA 92037.
  • Ganji S; Sanford-Burnham Medical Research Institute, La Jolla, CA 92037.
  • Zou J; Sanford-Burnham Medical Research Institute, La Jolla, CA 92037.
  • Pass I; Sanford-Burnham Medical Research Institute, La Jolla, CA 92037.
  • Narisawa S; Sanford-Burnham Medical Research Institute, La Jolla, CA 92037.
  • Iano FG; Sanford-Burnham Medical Research Institute, La Jolla, CA 92037.
  • Rosenstein C; Sanford-Burnham Medical Research Institute, La Jolla, CA 92037.
  • Cheltsov A; Sanford-Burnham Medical Research Institute, La Jolla, CA 92037.
  • Rascon J; Sanford-Burnham Medical Research Institute, La Jolla, CA 92037.
  • Hedrick M; Sanford-Burnham Medical Research Institute, La Jolla, CA 92037.
  • Gasior C; Sanford-Burnham Medical Research Institute, La Jolla, CA 92037.
  • Forster A; Sanford-Burnham Medical Research Institute, La Jolla, CA 92037.
  • Shi S; Sanford-Burnham Medical Research Institute, La Jolla, CA 92037.
  • Dahl R; Sanford-Burnham Medical Research Institute, La Jolla, CA 92037.
  • Vasile S; UCLA School of Medicine, Los Angeles, CA 90095.
  • Su Y; Sanford-Burnham Medical Research Institute, La Jolla, CA 92037.
  • Sergienko E; Sanford-Burnham Medical Research Institute, La Jolla, CA 92037.
  • Chung TDY; Sanford-Burnham Medical Research Institute, La Jolla, CA 92037.
  • Kaunitz J; UCLA School of Medicine, Los Angeles, CA 90095.
  • Hoylaerts MF; Department of Cardiovascular Sciences, Center for Molecular and Vascular Biology, University of Leuven, Leuven, Belgium.
  • Pinkerton AB; Sanford-Burnham Medical Research Institute, La Jolla, CA 92037.
  • Millán JL; Sanford-Burnham Medical Research Institute, La Jolla, CA 92037.
Bioorg Med Chem Lett ; 24(3): 1000-1004, 2014 Feb 01.
Article em En | MEDLINE | ID: mdl-24412070

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Sulfonamidas / Fosfatase Alcalina / Acetanilidas Tipo de estudo: Diagnostic_studies / Screening_studies Limite: Animals / Humans Idioma: En Revista: Bioorg Med Chem Lett Ano de publicação: 2014 Tipo de documento: Article

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Sulfonamidas / Fosfatase Alcalina / Acetanilidas Tipo de estudo: Diagnostic_studies / Screening_studies Limite: Animals / Humans Idioma: En Revista: Bioorg Med Chem Lett Ano de publicação: 2014 Tipo de documento: Article