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Orally bioavailable factor Xa inhibitors containing alpha-substituted gem-dimethyl P4 moieties.
Orwat, Michael J; Qiao, Jennifer X; He, Kan; Rendina, Alan R; Luettgen, Joseph M; Rossi, Karen A; Xin, Baomin; Knabb, Robert M; Wexler, Ruth R; Lam, Patrick Y S; Pinto, Donald J P.
Afiliação
  • Orwat MJ; Bristol-Myers Squibb Company, Research and Development, PO Box 4000, Princeton, NJ 08543-4000, USA. Electronic address: michael.orwat@bms.com.
  • Qiao JX; Bristol-Myers Squibb Company, Research and Development, PO Box 4000, Princeton, NJ 08543-4000, USA.
  • He K; Bristol-Myers Squibb Company, Research and Development, PO Box 4000, Princeton, NJ 08543-4000, USA.
  • Rendina AR; Bristol-Myers Squibb Company, Research and Development, PO Box 4000, Princeton, NJ 08543-4000, USA.
  • Luettgen JM; Bristol-Myers Squibb Company, Research and Development, PO Box 4000, Princeton, NJ 08543-4000, USA.
  • Rossi KA; Bristol-Myers Squibb Company, Research and Development, PO Box 4000, Princeton, NJ 08543-4000, USA.
  • Xin B; Bristol-Myers Squibb Company, Research and Development, PO Box 4000, Princeton, NJ 08543-4000, USA.
  • Knabb RM; Bristol-Myers Squibb Company, Research and Development, PO Box 4000, Princeton, NJ 08543-4000, USA.
  • Wexler RR; Bristol-Myers Squibb Company, Research and Development, PO Box 4000, Princeton, NJ 08543-4000, USA.
  • Lam PY; Bristol-Myers Squibb Company, Research and Development, PO Box 4000, Princeton, NJ 08543-4000, USA.
  • Pinto DJ; Bristol-Myers Squibb Company, Research and Development, PO Box 4000, Princeton, NJ 08543-4000, USA.
Bioorg Med Chem Lett ; 24(15): 3341-5, 2014 Aug 01.
Article em En | MEDLINE | ID: mdl-24951330

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Pirazóis / Piridonas / Fator Xa / Inibidores do Fator Xa Tipo de estudo: Prognostic_studies Limite: Animals / Humans Idioma: En Revista: Bioorg Med Chem Lett Ano de publicação: 2014 Tipo de documento: Article

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Pirazóis / Piridonas / Fator Xa / Inibidores do Fator Xa Tipo de estudo: Prognostic_studies Limite: Animals / Humans Idioma: En Revista: Bioorg Med Chem Lett Ano de publicação: 2014 Tipo de documento: Article