Your browser doesn't support javascript.
loading
A potentiator of orthosteric ligand activity at GLP-1R acts via covalent modification.
Nolte, Whitney M; Fortin, Jean-Philippe; Stevens, Benjamin D; Aspnes, Gary E; Griffith, David A; Hoth, Lise R; Ruggeri, Roger B; Mathiowetz, Alan M; Limberakis, Chris; Hepworth, David; Carpino, Philip A.
Afiliação
  • Nolte WM; Worldwide Medicinal Chemistry, Pfizer PharmaTherapeutics Research and Development, Cambridge, Massachusetts, USA.
  • Fortin JP; Cardiovascular and Metabolic Diseases Research Unit, Pfizer PharmaTherapeutics Research and Development, Cambridge, Massachusetts, USA.
  • Stevens BD; Worldwide Medicinal Chemistry, Pfizer PharmaTherapeutics Research and Development, Cambridge, Massachusetts, USA.
  • Aspnes GE; Worldwide Medicinal Chemistry, Pfizer PharmaTherapeutics Research and Development, Groton, Connecticut, USA.
  • Griffith DA; Worldwide Medicinal Chemistry, Pfizer PharmaTherapeutics Research and Development, Cambridge, Massachusetts, USA.
  • Hoth LR; Structural Biology and Biophysics Group, Center for Chemistry Innovation and Excellence, Worldwide Medicinal Chemistry, Pfizer PharmaTherapeutics Research and Development, Groton, Connecticut, USA.
  • Ruggeri RB; Worldwide Medicinal Chemistry, Pfizer PharmaTherapeutics Research and Development, Cambridge, Massachusetts, USA.
  • Mathiowetz AM; Worldwide Medicinal Chemistry, Pfizer PharmaTherapeutics Research and Development, Cambridge, Massachusetts, USA.
  • Limberakis C; Worldwide Medicinal Chemistry, Pfizer PharmaTherapeutics Research and Development, Groton, Connecticut, USA.
  • Hepworth D; Worldwide Medicinal Chemistry, Pfizer PharmaTherapeutics Research and Development, Cambridge, Massachusetts, USA.
  • Carpino PA; Worldwide Medicinal Chemistry, Pfizer PharmaTherapeutics Research and Development, Cambridge, Massachusetts, USA.
Nat Chem Biol ; 10(8): 629-31, 2014 Aug.
Article em En | MEDLINE | ID: mdl-24997604

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Pirimidinas / Receptores de Glucagon Limite: Animals / Humans Idioma: En Revista: Nat Chem Biol Ano de publicação: 2014 Tipo de documento: Article

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Pirimidinas / Receptores de Glucagon Limite: Animals / Humans Idioma: En Revista: Nat Chem Biol Ano de publicação: 2014 Tipo de documento: Article