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Synthesis and structure-activity-relationship studies of thiazolidinediones as antiplasmodial inhibitors of the Plasmodium falciparum cysteine protease falcipain-2.
Sharma, Rajni Kant; Younis, Yassir; Mugumbate, Grace; Njoroge, Mathew; Gut, Jiri; Rosenthal, Philip J; Chibale, Kelly.
Afiliação
  • Sharma RK; Department of Chemistry, University of Cape Town, Rondebosch 7701, South Africa.
  • Younis Y; Department of Chemistry, University of Cape Town, Rondebosch 7701, South Africa.
  • Mugumbate G; Department of Chemistry, University of Cape Town, Rondebosch 7701, South Africa.
  • Njoroge M; Department of Chemistry, University of Cape Town, Rondebosch 7701, South Africa.
  • Gut J; Department of Medicine, University of California, San Francisco, CA 94143, USA.
  • Rosenthal PJ; Department of Medicine, University of California, San Francisco, CA 94143, USA.
  • Chibale K; Department of Chemistry, University of Cape Town, Rondebosch 7701, South Africa; Institute of Infectious Disease and Molecular Medicine, University of Cape Town, Rondebosch 7701, South Africa; South African Medical Research Council, Drug Discovery and Development Unit, University of Cape Town, Ronde
Eur J Med Chem ; 90: 507-18, 2015 Jan 27.
Article em En | MEDLINE | ID: mdl-25486422

Texto completo: 1 Coleções: 01-internacional Contexto em Saúde: 3_ND Base de dados: MEDLINE Assunto principal: Plasmodium falciparum / Cisteína Endopeptidases / Inibidores de Cisteína Proteinase / Tiazolidinedionas / Antimaláricos Idioma: En Revista: Eur J Med Chem Ano de publicação: 2015 Tipo de documento: Article

Texto completo: 1 Coleções: 01-internacional Contexto em Saúde: 3_ND Base de dados: MEDLINE Assunto principal: Plasmodium falciparum / Cisteína Endopeptidases / Inibidores de Cisteína Proteinase / Tiazolidinedionas / Antimaláricos Idioma: En Revista: Eur J Med Chem Ano de publicação: 2015 Tipo de documento: Article