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The 8-Pyrrole-Benzothiazinones Are Noncovalent Inhibitors of DprE1 from Mycobacterium tuberculosis.
Makarov, Vadim; Neres, João; Hartkoorn, Ruben C; Ryabova, Olga B; Kazakova, Elena; Sarkan, Michal; Huszár, Stanislav; Piton, Jérémie; Kolly, Gaëlle S; Vocat, Anthony; Conroy, Trent M; Mikusová, Katarína; Cole, Stewart T.
Afiliação
  • Makarov V; More Medicines for Tuberculosis Consortium‡ A. N. Bakh Institute of Biochemistry, Russian Academy of Sciences, Moscow, Russia.
  • Neres J; More Medicines for Tuberculosis Consortium‡ Global Health Institute, Ecole Polytechnique Fédérale de Lausanne, Lausanne, Switzerland.
  • Hartkoorn RC; More Medicines for Tuberculosis Consortium‡ Global Health Institute, Ecole Polytechnique Fédérale de Lausanne, Lausanne, Switzerland.
  • Ryabova OB; More Medicines for Tuberculosis Consortium‡ A. N. Bakh Institute of Biochemistry, Russian Academy of Sciences, Moscow, Russia.
  • Kazakova E; More Medicines for Tuberculosis Consortium‡ A. N. Bakh Institute of Biochemistry, Russian Academy of Sciences, Moscow, Russia.
  • Sarkan M; More Medicines for Tuberculosis Consortium‡ Department of Biochemistry, Faculty of Natural Sciences, Comenius University in Bratislava, Bratislava, Slovakia.
  • Huszár S; More Medicines for Tuberculosis Consortium‡ Department of Biochemistry, Faculty of Natural Sciences, Comenius University in Bratislava, Bratislava, Slovakia.
  • Piton J; More Medicines for Tuberculosis Consortium‡ Global Health Institute, Ecole Polytechnique Fédérale de Lausanne, Lausanne, Switzerland.
  • Kolly GS; More Medicines for Tuberculosis Consortium‡ Global Health Institute, Ecole Polytechnique Fédérale de Lausanne, Lausanne, Switzerland.
  • Vocat A; More Medicines for Tuberculosis Consortium‡ Global Health Institute, Ecole Polytechnique Fédérale de Lausanne, Lausanne, Switzerland.
  • Conroy TM; More Medicines for Tuberculosis Consortium‡ Global Health Institute, Ecole Polytechnique Fédérale de Lausanne, Lausanne, Switzerland.
  • Mikusová K; More Medicines for Tuberculosis Consortium‡ Department of Biochemistry, Faculty of Natural Sciences, Comenius University in Bratislava, Bratislava, Slovakia.
  • Cole ST; More Medicines for Tuberculosis Consortium‡ Global Health Institute, Ecole Polytechnique Fédérale de Lausanne, Lausanne, Switzerland stewart.cole@epfl.ch.
Antimicrob Agents Chemother ; 59(8): 4446-52, 2015 Aug.
Article em En | MEDLINE | ID: mdl-25987616

Texto completo: 1 Coleções: 01-internacional Contexto em Saúde: 2_ODS3 / 3_ND Base de dados: MEDLINE Assunto principal: Piperazinas / Piridinas / Pirróis / Compostos de Espiro / Tiazinas / Proteínas de Bactérias / Oxirredutases do Álcool / Mycobacterium tuberculosis Limite: Animals / Humans / Male Idioma: En Revista: Antimicrob Agents Chemother Ano de publicação: 2015 Tipo de documento: Article

Texto completo: 1 Coleções: 01-internacional Contexto em Saúde: 2_ODS3 / 3_ND Base de dados: MEDLINE Assunto principal: Piperazinas / Piridinas / Pirróis / Compostos de Espiro / Tiazinas / Proteínas de Bactérias / Oxirredutases do Álcool / Mycobacterium tuberculosis Limite: Animals / Humans / Male Idioma: En Revista: Antimicrob Agents Chemother Ano de publicação: 2015 Tipo de documento: Article