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Synthesis, biological characterisation and structure activity relationships of aromatic bisamidines active against Plasmodium falciparum.
Sauer, B; Skinner-Adams, T S; Bouchut, A; Chua, M J; Pierrot, C; Erdmann, F; Robaa, D; Schmidt, M; Khalife, J; Andrews, K T; Sippl, W.
Afiliação
  • Sauer B; Martin-Luther-University Halle-Wittenberg, Wolfgang-Langenbeck-Str. 4, 06120, Halle, Germany.
  • Skinner-Adams TS; Tropical Parasitology Lab, Eskitis Institute for Drug Discovery, Don Young Road, Griffith University, Nathan, Queensland, 4111, Australia.
  • Bouchut A; U1019-CNRS UMR 8204, Univ. Lille Nord de France, Institut Pasteur de Lille, 1, Rue du professeur Calmette, 59019, Lille, France.
  • Chua MJ; Tropical Parasitology Lab, Eskitis Institute for Drug Discovery, Don Young Road, Griffith University, Nathan, Queensland, 4111, Australia.
  • Pierrot C; U1019-CNRS UMR 8204, Univ. Lille Nord de France, Institut Pasteur de Lille, 1, Rue du professeur Calmette, 59019, Lille, France.
  • Erdmann F; Martin-Luther-University Halle-Wittenberg, Wolfgang-Langenbeck-Str. 4, 06120, Halle, Germany.
  • Robaa D; Martin-Luther-University Halle-Wittenberg, Wolfgang-Langenbeck-Str. 4, 06120, Halle, Germany.
  • Schmidt M; Martin-Luther-University Halle-Wittenberg, Wolfgang-Langenbeck-Str. 4, 06120, Halle, Germany.
  • Khalife J; U1019-CNRS UMR 8204, Univ. Lille Nord de France, Institut Pasteur de Lille, 1, Rue du professeur Calmette, 59019, Lille, France.
  • Andrews KT; Tropical Parasitology Lab, Eskitis Institute for Drug Discovery, Don Young Road, Griffith University, Nathan, Queensland, 4111, Australia.
  • Sippl W; Martin-Luther-University Halle-Wittenberg, Wolfgang-Langenbeck-Str. 4, 06120, Halle, Germany. Electronic address: wolfgang.sippl@pharmazie.uni-halle.de.
Eur J Med Chem ; 127: 22-40, 2017 Feb 15.
Article em En | MEDLINE | ID: mdl-28038325

Texto completo: 1 Coleções: 01-internacional Contexto em Saúde: 3_ND Base de dados: MEDLINE Assunto principal: Plasmodium falciparum / Furanos / Antimaláricos Limite: Humans Idioma: En Revista: Eur J Med Chem Ano de publicação: 2017 Tipo de documento: Article

Texto completo: 1 Coleções: 01-internacional Contexto em Saúde: 3_ND Base de dados: MEDLINE Assunto principal: Plasmodium falciparum / Furanos / Antimaláricos Limite: Humans Idioma: En Revista: Eur J Med Chem Ano de publicação: 2017 Tipo de documento: Article