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An Intracellular Allosteric Modulator Binding Pocket in SK2 Ion Channels Is Shared by Multiple Chemotypes.
Cho, Lily T-Y; Alexandrou, Aristos J; Torella, Rubben; Knafels, John; Hobbs, Jake; Taylor, Toni; Loucif, Alex; Konopacka, Agnieszka; Bell, Sigourney; Stevens, Edward B; Pandit, Jay; Horst, Reto; Withka, Jane M; Pryde, David C; Liu, Shenping; Young, Gareth T.
Afiliação
  • Cho LT; Pfizer Neuroscience and Pain Research Unit, Granta Park, Great Abington, Cambridge CB21 6GS, UK.
  • Alexandrou AJ; Pfizer Neuroscience and Pain Research Unit, Granta Park, Great Abington, Cambridge CB21 6GS, UK.
  • Torella R; Pfizer Worldwide Medicinal Chemistry, Neuroscience and Pain Research Unit, Granta Park, Great Abington, Cambridge CB21 6GS, UK.
  • Knafels J; Pfizer Structural Biology and Biophysics, Groton, Eastern Point Road, Groton, CT 06340, USA.
  • Hobbs J; Pfizer Neuroscience and Pain Research Unit, Granta Park, Great Abington, Cambridge CB21 6GS, UK.
  • Taylor T; Pfizer Neuroscience and Pain Research Unit, Granta Park, Great Abington, Cambridge CB21 6GS, UK.
  • Loucif A; Pfizer Neuroscience and Pain Research Unit, Granta Park, Great Abington, Cambridge CB21 6GS, UK.
  • Konopacka A; Pfizer Neuroscience and Pain Research Unit, Granta Park, Great Abington, Cambridge CB21 6GS, UK.
  • Bell S; Pfizer Neuroscience and Pain Research Unit, Granta Park, Great Abington, Cambridge CB21 6GS, UK.
  • Stevens EB; Pfizer Neuroscience and Pain Research Unit, Granta Park, Great Abington, Cambridge CB21 6GS, UK.
  • Pandit J; Pfizer Structural Biology and Biophysics, Groton, Eastern Point Road, Groton, CT 06340, USA.
  • Horst R; Pfizer Structural Biology and Biophysics, Groton, Eastern Point Road, Groton, CT 06340, USA.
  • Withka JM; Pfizer Structural Biology and Biophysics, Groton, Eastern Point Road, Groton, CT 06340, USA.
  • Pryde DC; Pfizer Worldwide Medicinal Chemistry, Neuroscience and Pain Research Unit, Granta Park, Great Abington, Cambridge CB21 6GS, UK.
  • Liu S; Pfizer Structural Biology and Biophysics, Groton, Eastern Point Road, Groton, CT 06340, USA. Electronic address: shenping.liu@pfizer.com.
  • Young GT; Pfizer Neuroscience and Pain Research Unit, Granta Park, Great Abington, Cambridge CB21 6GS, UK. Electronic address: gareth.8.young@gsk.com.
Structure ; 26(4): 533-544.e3, 2018 04 03.
Article em En | MEDLINE | ID: mdl-29576321

Texto completo: 1 Coleções: 01-internacional Contexto em Saúde: 3_ND Base de dados: MEDLINE Assunto principal: Oximas / Pirazóis / Pirimidinas / Calmodulina / Riluzol / Canais de Potássio Ativados por Cálcio de Condutância Baixa / Indóis Tipo de estudo: Prognostic_studies Limite: Humans Idioma: En Revista: Structure Ano de publicação: 2018 Tipo de documento: Article

Texto completo: 1 Coleções: 01-internacional Contexto em Saúde: 3_ND Base de dados: MEDLINE Assunto principal: Oximas / Pirazóis / Pirimidinas / Calmodulina / Riluzol / Canais de Potássio Ativados por Cálcio de Condutância Baixa / Indóis Tipo de estudo: Prognostic_studies Limite: Humans Idioma: En Revista: Structure Ano de publicação: 2018 Tipo de documento: Article