Discovery of 2-aminoimidazole and 2-amino imidazolyl-thiazoles as non-xanthine human adenosine A<sub>3</sub> receptor antagonists: SAR and molecular modeling studies.

Pandya, Amit N; Baraiya, Arshi B; Jalani, Hitesh B; Pandya, Dhaivat; Kaila, Jitendra C; Kachler, Sonja; Salmaso, Veronica; Moro, Stefano; Klotz, Karl-Norbert; Vasu, Kamala K

Discovery of 2-aminoimidazole and 2-amino imidazolyl-thiazoles as non-xanthine human adenosine A₃ receptor antagonists: SAR and molecular modeling studies.

Pandya, Amit N; Baraiya, Arshi B; Jalani, Hitesh B; Pandya, Dhaivat; Kaila, Jitendra C; Kachler, Sonja; Salmaso, Veronica; Moro, Stefano; Klotz, Karl-Norbert; Vasu, Kamala K.

Afiliação

Pandya AN; Department of Medicinal Chemistry , B. V. Patel Pharmaceutical Education and Research Development (PERD) Centre , Sarkej-Gandhinagar Highway, Thaltej , Ahmedabad 380e054 , Gujarat , India . Email: kamalav@perdcentre.com ; Email: kamkva@gmail.com.
Baraiya AB; Department of Medicinal Chemistry , B. V. Patel Pharmaceutical Education and Research Development (PERD) Centre , Sarkej-Gandhinagar Highway, Thaltej , Ahmedabad 380e054 , Gujarat , India . Email: kamalav@perdcentre.com ; Email: kamkva@gmail.com.
Jalani HB; Department of Medicinal Chemistry , B. V. Patel Pharmaceutical Education and Research Development (PERD) Centre , Sarkej-Gandhinagar Highway, Thaltej , Ahmedabad 380e054 , Gujarat , India . Email: kamalav@perdcentre.com ; Email: kamkva@gmail.com.
Pandya D; Department of Medicinal Chemistry , B. V. Patel Pharmaceutical Education and Research Development (PERD) Centre , Sarkej-Gandhinagar Highway, Thaltej , Ahmedabad 380e054 , Gujarat , India . Email: kamalav@perdcentre.com ; Email: kamkva@gmail.com.
Kaila JC; Department of Medicinal Chemistry , B. V. Patel Pharmaceutical Education and Research Development (PERD) Centre , Sarkej-Gandhinagar Highway, Thaltej , Ahmedabad 380e054 , Gujarat , India . Email: kamalav@perdcentre.com ; Email: kamkva@gmail.com.
Kachler S; Institut für Pharmakologie und Toxikologie , Julius-Maximilians-Universität Würzburg , Germany.
Salmaso V; Molecular Modeling Section (MMS) , Dipartimento di Scienze Farmaceutiche , Università degli Studi di Padova , via Marzolo 5 , 35131 Padova , Italy.
Moro S; Molecular Modeling Section (MMS) , Dipartimento di Scienze Farmaceutiche , Università degli Studi di Padova , via Marzolo 5 , 35131 Padova , Italy.
Klotz KN; Institut für Pharmakologie und Toxikologie , Julius-Maximilians-Universität Würzburg , Germany.
Vasu KK; Department of Medicinal Chemistry , B. V. Patel Pharmaceutical Education and Research Development (PERD) Centre , Sarkej-Gandhinagar Highway, Thaltej , Ahmedabad 380e054 , Gujarat , India . Email: kamalav@perdcentre.com ; Email: kamkva@gmail.com.

Medchemcomm ; 9(4): 676-684, 2018 Apr 01.

Article em En | MEDLINE | ID: mdl-30108958

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Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Idioma: En Revista: Medchemcomm Ano de publicação: 2018 Tipo de documento: Article

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Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Idioma: En Revista: Medchemcomm Ano de publicação: 2018 Tipo de documento: Article