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Synthesis and evaluation of Re/99mTc(I) complexes bearing a somatostatin receptor-targeting antagonist and labeled via a novel [N,S,O] clickable bifunctional chelating agent.
Radford, Lauren L; Papagiannopoulou, Dionysia; Gallazzi, Fabio; Berendzen, Ashley; Watkinson, Lisa; Carmack, Terry; Lewis, Michael R; Jurisson, Silvia S; Hennkens, Heather M.
Afiliação
  • Radford LL; Department of Chemistry, University of Missouri, 601 S. College Ave., Columbia, MO 65211, USA.
  • Papagiannopoulou D; School of Pharmacy, Aristotle University of Thessaloniki, 54124 Thessaloniki, Greece.
  • Gallazzi F; Department of Chemistry, University of Missouri, 601 S. College Ave., Columbia, MO 65211, USA; Molecular Interaction Core, University of Missouri, 601 S. College Ave., Columbia, MO 65211, USA.
  • Berendzen A; Research Service, Harry S. Truman Memorial Veterans' Hospital, 800 Hospital Dr., Columbia, MO 65212, USA.
  • Watkinson L; Research Service, Harry S. Truman Memorial Veterans' Hospital, 800 Hospital Dr., Columbia, MO 65212, USA.
  • Carmack T; Research Service, Harry S. Truman Memorial Veterans' Hospital, 800 Hospital Dr., Columbia, MO 65212, USA.
  • Lewis MR; Research Service, Harry S. Truman Memorial Veterans' Hospital, 800 Hospital Dr., Columbia, MO 65212, USA; Department of Veterinary Medicine and Surgery, University of Missouri, 900 E Campus Dr., Columbia, MO 65211, USA.
  • Jurisson SS; Department of Chemistry, University of Missouri, 601 S. College Ave., Columbia, MO 65211, USA.
  • Hennkens HM; Department of Chemistry, University of Missouri, 601 S. College Ave., Columbia, MO 65211, USA; University of Missouri Research Reactor Center, 1513 Research Park Dr., Columbia, MO 65211, USA. Electronic address: HennkensH@missouri.edu.
Bioorg Med Chem ; 27(3): 492-501, 2019 02 01.
Article em En | MEDLINE | ID: mdl-30594453

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Compostos Organometálicos / Rênio / Quelantes / Tecnécio / Receptores de Somatostatina / Compostos Radiofarmacêuticos Limite: Animals Idioma: En Revista: Bioorg Med Chem Ano de publicação: 2019 Tipo de documento: Article

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Compostos Organometálicos / Rênio / Quelantes / Tecnécio / Receptores de Somatostatina / Compostos Radiofarmacêuticos Limite: Animals Idioma: En Revista: Bioorg Med Chem Ano de publicação: 2019 Tipo de documento: Article