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3D QSAR-based design and liquid phase combinatorial synthesis of 1,2-disubstituted benzimidazole-5-carboxylic acid and 3-substituted-5H-benzimidazo[1,2-d][1,4]benzodiazepin-6(7H)-one derivatives as anti-mycobacterial agents.
Sitwala, Nikum D; Vyas, Vivek K; Gedia, Piyush; Patel, Kinjal; Bouzeyen, Rania; Kidwai, Saqib; Singh, Ramandeep; Ghate, Manjunath D.
Afiliação
  • Sitwala ND; Department of Pharmaceutical Chemistry, Institute of Pharmacy , Nirma University , Ahmedabad 382481 , Gujarat , India . Email: manjunath.ghate@nirmauni.ac.in.
  • Vyas VK; Department of Pharmaceutical Chemistry, Institute of Pharmacy , Nirma University , Ahmedabad 382481 , Gujarat , India . Email: manjunath.ghate@nirmauni.ac.in.
  • Gedia P; Department of Pharmaceutical Chemistry, Institute of Pharmacy , Nirma University , Ahmedabad 382481 , Gujarat , India . Email: manjunath.ghate@nirmauni.ac.in.
  • Patel K; Department of Pharmaceutical Chemistry, Institute of Pharmacy , Nirma University , Ahmedabad 382481 , Gujarat , India . Email: manjunath.ghate@nirmauni.ac.in.
  • Bouzeyen R; Institut Pasteur de Tunis , LTCII, LR11 IPT02 , Tunis , 1002 , Tunisia.
  • Kidwai S; Université Tunis El Manar , Tunis , 1068 , Tunisia.
  • Singh R; Tuberculosis Research Laboratory , Vaccine and Infectious Disease Research Centre , Translational Health Science and Technology Institute , Faridabad-Gurugram Expressway , Haryana , India.
  • Ghate MD; Tuberculosis Research Laboratory , Vaccine and Infectious Disease Research Centre , Translational Health Science and Technology Institute , Faridabad-Gurugram Expressway , Haryana , India.
Medchemcomm ; 10(5): 817-827, 2019 May 01.
Article em En | MEDLINE | ID: mdl-31293724

Texto completo: 1 Coleções: 01-internacional Contexto em Saúde: 3_ND Base de dados: MEDLINE Tipo de estudo: Prognostic_studies Idioma: En Revista: Medchemcomm Ano de publicação: 2019 Tipo de documento: Article

Texto completo: 1 Coleções: 01-internacional Contexto em Saúde: 3_ND Base de dados: MEDLINE Tipo de estudo: Prognostic_studies Idioma: En Revista: Medchemcomm Ano de publicação: 2019 Tipo de documento: Article