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Design and synthesis of novel pyrrolo[2,3-b]pyridine derivatives targeting V600EBRAF.
Abdel-Maksoud, Mohammed S; Ali, Eslam M H; Ammar, Usama M; Mersal, Karim I; Yoo, Kyung Ho; Oh, Chang-Hyun.
Afiliação
  • Abdel-Maksoud MS; Medicinal &Pharmaceutical Chemistry Department, Pharmaceutical and Drug Industries Research Division, National Research Centre (NRC ID: 60014618), Dokki, Giza 12622, Egypt.
  • Ali EMH; Center for Biomaterials, Korea Institute of Science & Technology (KIST School), Seoul, Seongbuk-gu 02792, Republic of Korea; University of Science & Technology (UST), Daejeon, Yuseong-gu 34113, Republic of Korea; Pharmaceutical Chemistry Department, Faculty of Pharmacy, Modern University of
  • Ammar UM; Center for Biomaterials, Korea Institute of Science & Technology (KIST School), Seoul, Seongbuk-gu 02792, Republic of Korea; University of Science & Technology (UST), Daejeon, Yuseong-gu 34113, Republic of Korea; Pharmaceutical Chemistry Department, Faculty of Pharmacy, Ahram Canadian Univer
  • Mersal KI; Center for Biomaterials, Korea Institute of Science & Technology (KIST School), Seoul, Seongbuk-gu 02792, Republic of Korea; University of Science & Technology (UST), Daejeon, Yuseong-gu 34113, Republic of Korea.
  • Yoo KH; Chemical Kinomics Research Center, Korea Institute of Science and Technology, Seoul, Republic of Korea.
  • Oh CH; Center for Biomaterials, Korea Institute of Science & Technology (KIST School), Seoul, Seongbuk-gu 02792, Republic of Korea; University of Science & Technology (UST), Daejeon, Yuseong-gu 34113, Republic of Korea. Electronic address: choh@kist.re.kr.
Bioorg Med Chem ; 28(11): 115493, 2020 06 01.
Article em En | MEDLINE | ID: mdl-32340792

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Piridinas / Pirróis / Desenho de Fármacos / Proteínas Proto-Oncogênicas B-raf / Inibidores de Proteínas Quinases / Antineoplásicos Limite: Humans Idioma: En Revista: Bioorg Med Chem Ano de publicação: 2020 Tipo de documento: Article

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Piridinas / Pirróis / Desenho de Fármacos / Proteínas Proto-Oncogênicas B-raf / Inibidores de Proteínas Quinases / Antineoplásicos Limite: Humans Idioma: En Revista: Bioorg Med Chem Ano de publicação: 2020 Tipo de documento: Article