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Development of small-molecule inhibitors of fatty acyl-AMP and fatty acyl-CoA ligases in Mycobacterium tuberculosis.
Baran, Marzena; Grimes, Kimberly D; Sibbald, Paul A; Fu, Peng; Boshoff, Helena I M; Wilson, Daniel J; Aldrich, Courtney C.
Afiliação
  • Baran M; Department of Medicinal Chemistry, University of Minnesota, 8-101 WDH, 308 Harvard Street SE, Minneapolis, MN, 55455, United States.
  • Grimes KD; Center for Drug Design, Academic Health Center, University of Minnesota, Minneapolis, MN, 55455, United States.
  • Sibbald PA; Center for Drug Design, Academic Health Center, University of Minnesota, Minneapolis, MN, 55455, United States.
  • Fu P; Center for Drug Design, Academic Health Center, University of Minnesota, Minneapolis, MN, 55455, United States.
  • Boshoff HIM; Tuberculosis Research Section, National Institute of Allergy and Infectious Diseases, Bethesda, MD, 20892, United States.
  • Wilson DJ; Center for Drug Design, Academic Health Center, University of Minnesota, Minneapolis, MN, 55455, United States.
  • Aldrich CC; Department of Medicinal Chemistry, University of Minnesota, 8-101 WDH, 308 Harvard Street SE, Minneapolis, MN, 55455, United States; Center for Drug Design, Academic Health Center, University of Minnesota, Minneapolis, MN, 55455, United States. Electronic address: aldri015@umn.edu.
Eur J Med Chem ; 201: 112408, 2020 Sep 01.
Article em En | MEDLINE | ID: mdl-32574901

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Adenosina / Coenzima A Ligases / Inibidores Enzimáticos / Mycobacterium tuberculosis / Antituberculosos Limite: Animals Idioma: En Revista: Eur J Med Chem Ano de publicação: 2020 Tipo de documento: Article

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Adenosina / Coenzima A Ligases / Inibidores Enzimáticos / Mycobacterium tuberculosis / Antituberculosos Limite: Animals Idioma: En Revista: Eur J Med Chem Ano de publicação: 2020 Tipo de documento: Article