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Synthesis, biological evaluation and in silico modeling of novel pan-genotypic NS5A inhibitors.
Ivashchenko, Andrey A; Ivanenkov, Yan A; Aladinskiy, Vladimir A; Karapetian, Ruben N; Koryakova, Angela G; Ryakhovskiy, Alexey A; Mitkin, Oleg D; Kravchenko, Dmitry V; Savchuk, Nikolai P; Zagribelnyy, Bogdan A; Ivashchenko, Alexander V.
Afiliação
  • Ivashchenko AA; Chemical Diversity Research Institute, Rabochaya St. 2a, Khimki, Moscow Region 141401, Russia; ChemDiv, 6605 Nancy Ridge Drive San Diego, CA 92121, United States; Moscow Institute of Physics and Technology (State University), 9 Institutskiy lane, Dolgoprudny City, Moscow Region 141700, Russia.
  • Ivanenkov YA; ChemDiv, 6605 Nancy Ridge Drive San Diego, CA 92121, United States; Institute of Biochemistry and Genetics Russian Academy of Science (IBG RAS) Ufa Scientific Centre, Ufa, Russia. Electronic address: yai@chemdiv.com.
  • Aladinskiy VA; Moscow Institute of Physics and Technology (State University), 9 Institutskiy lane, Dolgoprudny City, Moscow Region 141700, Russia.
  • Karapetian RN; Chemical Diversity Research Institute, Rabochaya St. 2a, Khimki, Moscow Region 141401, Russia.
  • Koryakova AG; Chemical Diversity Research Institute, Rabochaya St. 2a, Khimki, Moscow Region 141401, Russia.
  • Ryakhovskiy AA; Chemical Diversity Research Institute, Rabochaya St. 2a, Khimki, Moscow Region 141401, Russia.
  • Mitkin OD; Chemical Diversity Research Institute, Rabochaya St. 2a, Khimki, Moscow Region 141401, Russia.
  • Kravchenko DV; Chemical Diversity Research Institute, Rabochaya St. 2a, Khimki, Moscow Region 141401, Russia.
  • Savchuk NP; Chemical Diversity Research Institute, Rabochaya St. 2a, Khimki, Moscow Region 141401, Russia; Avisa Pharmaceuticals LLC, 1835 E. Hallandale Beach Blvd, #442, Hallandale Beach, Fl 33009, United States.
  • Zagribelnyy BA; Moscow Institute of Physics and Technology (State University), 9 Institutskiy lane, Dolgoprudny City, Moscow Region 141700, Russia.
  • Ivashchenko AV; Chemical Diversity Research Institute, Rabochaya St. 2a, Khimki, Moscow Region 141401, Russia; ChemDiv, 6605 Nancy Ridge Drive San Diego, CA 92121, United States; Avisa Pharmaceuticals LLC, 1835 E. Hallandale Beach Blvd, #442, Hallandale Beach, Fl 33009, United States.
Bioorg Med Chem ; 28(20): 115716, 2020 10 15.
Article em En | MEDLINE | ID: mdl-33069072

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Antivirais / Proteínas não Estruturais Virais / Hepacivirus / Imidazóis Tipo de estudo: Prognostic_studies Limite: Animals / Humans / Male Idioma: En Revista: Bioorg Med Chem Ano de publicação: 2020 Tipo de documento: Article

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Antivirais / Proteínas não Estruturais Virais / Hepacivirus / Imidazóis Tipo de estudo: Prognostic_studies Limite: Animals / Humans / Male Idioma: En Revista: Bioorg Med Chem Ano de publicação: 2020 Tipo de documento: Article