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Discovery of ZN-c3, a Highly Potent and Selective Wee1 Inhibitor Undergoing Evaluation in Clinical Trials for the Treatment of Cancer.
Huang, Peter Q; Boren, Brant C; Hegde, Sayee G; Liu, Hui; Unni, Aditya K; Abraham, Sunny; Hopkins, Chad D; Paliwal, Sunil; Samatar, Ahmed A; Li, Jiali; Bunker, Kevin D.
Afiliação
  • Huang PQ; Zentalis Pharmaceuticals, San Diego, California 92121, United States.
  • Boren BC; Zentalis Pharmaceuticals, San Diego, California 92121, United States.
  • Hegde SG; Zentalis Pharmaceuticals, San Diego, California 92121, United States.
  • Liu H; Zentalis Pharmaceuticals, San Diego, California 92121, United States.
  • Unni AK; Zentalis Pharmaceuticals, San Diego, California 92121, United States.
  • Abraham S; Zentalis Pharmaceuticals, San Diego, California 92121, United States.
  • Hopkins CD; Zentalis Pharmaceuticals, San Diego, California 92121, United States.
  • Paliwal S; Zentalis Pharmaceuticals, San Diego, California 92121, United States.
  • Samatar AA; Zentalis Pharmaceuticals, San Diego, California 92121, United States.
  • Li J; Zentalis Pharmaceuticals, San Diego, California 92121, United States.
  • Bunker KD; Zentalis Pharmaceuticals, San Diego, California 92121, United States.
J Med Chem ; 64(17): 13004-13024, 2021 09 09.
Article em En | MEDLINE | ID: mdl-34423975

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Proteínas Tirosina Quinases / Proteínas de Ciclo Celular / Descoberta de Drogas / Antineoplásicos Tipo de estudo: Prognostic_studies Limite: Animals / Humans / Male Idioma: En Revista: J Med Chem Ano de publicação: 2021 Tipo de documento: Article

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Proteínas Tirosina Quinases / Proteínas de Ciclo Celular / Descoberta de Drogas / Antineoplásicos Tipo de estudo: Prognostic_studies Limite: Animals / Humans / Male Idioma: En Revista: J Med Chem Ano de publicação: 2021 Tipo de documento: Article