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Macrocyclic peptides as allosteric inhibitors of nicotinamide N-methyltransferase (NNMT).
van Haren, Matthijs J; Zhang, Yurui; Thijssen, Vito; Buijs, Ned; Gao, Yongzhi; Mateuszuk, Lukasz; Fedak, Filip A; Kij, Agnieszka; Campagna, Roberto; Sartini, Davide; Emanuelli, Monica; Chlopicki, Stefan; Jongkees, Seino A K; Martin, Nathaniel I.
Afiliação
  • van Haren MJ; Biological Chemistry Group, Institute of Biology Leiden, Leiden University Sylviusweg 72 2333 BE Leiden The Netherlands n.i.martin@biology.leidenuniv.nl.
  • Zhang Y; Biological Chemistry Group, Institute of Biology Leiden, Leiden University Sylviusweg 72 2333 BE Leiden The Netherlands n.i.martin@biology.leidenuniv.nl.
  • Thijssen V; Chemical Biology & Drug Discovery Group, Utrecht Institute for Pharmaceutical Sciences Universiteitsweg 99 3584 CG Utrecht The Netherlands s.a.k.jongkees@vu.nl.
  • Buijs N; Biological Chemistry Group, Institute of Biology Leiden, Leiden University Sylviusweg 72 2333 BE Leiden The Netherlands n.i.martin@biology.leidenuniv.nl.
  • Gao Y; Biological Chemistry Group, Institute of Biology Leiden, Leiden University Sylviusweg 72 2333 BE Leiden The Netherlands n.i.martin@biology.leidenuniv.nl.
  • Mateuszuk L; Jagiellonian University, Jagiellonian Centre for Experimental Therapeutics (JCET) Bobrzynskiego 14 30-348 Krakow Poland.
  • Fedak FA; Jagiellonian University, Jagiellonian Centre for Experimental Therapeutics (JCET) Bobrzynskiego 14 30-348 Krakow Poland.
  • Kij A; Jagiellonian University, Jagiellonian Centre for Experimental Therapeutics (JCET) Bobrzynskiego 14 30-348 Krakow Poland.
  • Campagna R; Department of Clinical Sciences, Universitá Politecnica delle Marche Via Ranieri 65 60131 Ancona Italy.
  • Sartini D; Department of Clinical Sciences, Universitá Politecnica delle Marche Via Ranieri 65 60131 Ancona Italy.
  • Emanuelli M; Department of Clinical Sciences, Universitá Politecnica delle Marche Via Ranieri 65 60131 Ancona Italy.
  • Chlopicki S; Jagiellonian University, Jagiellonian Centre for Experimental Therapeutics (JCET) Bobrzynskiego 14 30-348 Krakow Poland.
  • Jongkees SAK; Jagiellonian University Medical College, Chair of Pharmacology Grzegorzecka 16 31-531 Krakow Poland.
  • Martin NI; Chemical Biology & Drug Discovery Group, Utrecht Institute for Pharmaceutical Sciences Universiteitsweg 99 3584 CG Utrecht The Netherlands s.a.k.jongkees@vu.nl.
RSC Chem Biol ; 2(5): 1546-1555, 2021 Oct 07.
Article em En | MEDLINE | ID: mdl-34704059

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Idioma: En Revista: RSC Chem Biol Ano de publicação: 2021 Tipo de documento: Article

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Idioma: En Revista: RSC Chem Biol Ano de publicação: 2021 Tipo de documento: Article